129029-23-8 | Ocaperidone

Packsize	Purity	Availability	Price	Discounted Price
1mg	97%	in stock	$34.00	$24.00
5mg	97%	in stock	$84.00	$59.00
10mg	97%	in stock	$126.00	$88.00
25mg	>98.0%(HPLC)	in stock	$164.00	$115.00

Description

• Catalog Number: AA44901
• Chemical Name: Ocaperidone
• CAS Number: 129029-23-8
• Molecular Formula: C24H25FN4O2
• Molecular Weight: 420.4793
• MDL Number: MFCD00866668
• SMILES: Fc1ccc2c(c1)onc2C1CCN(CC1)CCc1c(C)nc2n(c1=O)cccc2C

Computed Properties

• Complexity: 856
• Covalently-Bonded Unit Count: 1
• Heavy Atom Count: 31
• Hydrogen Bond Acceptor Count: 6
• Rotatable Bond Count: 4
• XLogP3: 3.3

Literature

• Efficacy of antipsychotic agents at human 5-HT(1A) receptors determined by [3H]WAY100,635 binding affinity ratios: relationship to efficacy for G-protein activation.

  European journal of pharmacology 20011005

• Agonistic properties of alniditan, sumatriptan and dihydroergotamine on human 5-HT1B and 5-HT1D receptors expressed in various mammalian cell lines.

  British journal of pharmacology 19980401

• 5-HT1A receptor activates Na+/H+ exchange in CHO-K1 cells through Gialpha2 and Gialpha3.

  The Journal of biological chemistry 19970321

• Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamine and [3H]alniditan.

  Molecular pharmacology 19961201