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Molecular cloning, characterization, and inhibition studies of a β-carbonic anhydrase from Malassezia globosa, a potential antidandruff target.
Journal of medicinal chemistry 20120412
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Cloning, characterization and sulfonamide inhibition studies of an α-carbonic anhydrase from the living fossil sponge Astrosclera willeyana.
Bioorganic & medicinal chemistry 20120215
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Inhibition studies of the β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium with sulfonamides and sulfamates.
Bioorganic & medicinal chemistry 20110815
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New bitter blocker discovered, study finds.
Journal of the American Dental Association (1939) 20110801
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Polymers of 2-methacryloyloxyethyl phosphorylcholine truly work as cell membrane mimic?
Colloids and surfaces. B, Biointerfaces 20110501
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A new β-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth.
Bioorganic & medicinal chemistry 20110201
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Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata.
Bioorganic & medicinal chemistry letters 20110115
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Probenecid inhibits the human bitter taste receptor TAS2R16 and suppresses bitter perception of salicin.
PloS one 20110101
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Interaction-dependent PCR: identification of ligand-target pairs from libraries of ligands and libraries of targets in a single solution-phase experiment.
Journal of the American Chemical Society 20101110
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Cloning, characterization, and inhibition studies of a beta-carbonic anhydrase from Brucella suis.
Journal of medicinal chemistry 20100311
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Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c.
Bioorganic & medicinal chemistry letters 20091201
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Carbonic anhydrase inhibitors. Inhibition studies of a coral secretory isoform by sulfonamides.
Bioorganic & medicinal chemistry 20090715
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Carbonic anhydrase inhibitors. Inhibition and homology modeling studies of the fungal beta-carbonic anhydrase from Candida albicans with sulfonamides.
Bioorganic & medicinal chemistry 20090701
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Titration calorimetry standards and the precision of isothermal titration calorimetry data.
International journal of molecular sciences 20090601
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Carbonic anhydrase inhibitors. Cloning, characterization, and inhibition studies of a new beta-carbonic anhydrase from Mycobacterium tuberculosis.
Journal of medicinal chemistry 20090514
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Ligand-directed tosyl chemistry for protein labeling in vivo.
Nature chemical biology 20090501
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Molecular cloning, characterization, and inhibition studies of the Rv1284 beta-carbonic anhydrase from Mycobacterium tuberculosis with sulfonamides and a sulfamate.
Journal of medicinal chemistry 20090423
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Carbonic anhydrase inhibitors: inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamates.
Bioorganic & medicinal chemistry 20090201
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Label-free determination of protein-ligand binding constants using mass spectrometry and validation using surface plasmon resonance and isothermal titration calorimetry.
Journal of molecular recognition : JMR 20090101
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Using ion channel-forming peptides to quantify protein-ligand interactions.
Journal of the American Chemical Society 20080130
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Carbonic anhydrase inhibitors: cloning, characterization, and inhibition studies of the cytosolic isozyme III with sulfonamides.
Bioorganic & medicinal chemistry 20071201
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Implementation of chemometric methodology in ACE: predictive investigation of protein-ligand binding.
Electrophoresis 20070801
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Carbonic anhydrase inhibitors: the beta-carbonic anhydrase from Helicobacter pylori is a new target for sulfonamide and sulfamate inhibitors.
Bioorganic & medicinal chemistry letters 20070701
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Anti-mycobacterial activity of a bis-sulfonamide.
Bioorganic & medicinal chemistry letters 20070301
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Carbonic anhydrase inhibitors. DNA cloning, characterization, and inhibition studies of the human secretory isoform VI, a new target for sulfonamide and sulfamate inhibitors.
Journal of medicinal chemistry 20070125
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Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
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Carbonic anhydrase inhibitors: cloning and sulfonamide inhibition studies of a carboxyterminal truncated alpha-carbonic anhydrase from Helicobacter pylori.
Bioorganic & medicinal chemistry letters 20060415
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Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs.
Journal of medicinal chemistry 20060323
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Synthesis and structure-activity relationships of novel benzene sulfonamides with potent binding affinity for bovine carbonic anhydrase II.
Bioorganic & medicinal chemistry letters 20051215
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Carbonic anhydrase inhibitors. The mitochondrial isozyme VB as a new target for sulfonamide and sulfamate inhibitors.
Journal of medicinal chemistry 20051201
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Carbonic anhydrase inhibitors: inhibition of the transmembrane isozyme XIV with sulfonamides.
Bioorganic & medicinal chemistry letters 20050901
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Carbonic anhydrase inhibitors. Inhibition of the transmembrane isozyme XII with sulfonamides-a new target for the design of antitumor and antiglaucoma drugs?
Bioorganic & medicinal chemistry letters 20050215
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Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isozyme VII with aromatic and heterocyclic sulfonamides.
Bioorganic & medicinal chemistry letters 20050215
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Carbonic anhydrase inhibitors: inhibition of human cytosolic isozyme II and mitochondrial isozyme V with a series of benzene sulfonamide derivatives.
Bioorganic & medicinal chemistry letters 20041115
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Synthesis of 4,5-diaryl-1H-pyrazole-3-ol derivatives as potential COX-2 inhibitors.
The Journal of organic chemistry 20041015
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Carbonic anhydrase inhibitors: the first QSAR study on inhibition of tumor-associated isoenzyme IX with aromatic and heterocyclic sulfonamides.
Bioorganic & medicinal chemistry letters 20040621
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The ABRF-MIRG'02 study: assembly state, thermodynamic, and kinetic analysis of an enzyme/inhibitor interaction.
Journal of biomolecular techniques : JBT 20031201
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Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with a bis-sulfonamide-two heads are better than one?
Bioorganic & medicinal chemistry letters 20030818
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Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides.
Bioorganic & medicinal chemistry letters 20030324
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Direct comparison of binding equilibrium, thermodynamic, and rate constants determined by surface- and solution-based biophysical methods.
Protein science : a publication of the Protein Society 20020501
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Back to basics.
Genome biology 20020101
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Biodegradation of p-toluenesulphonamide by a Pseudomonas sp.
FEMS microbiology letters 20011113
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Carbonic anhydrase inhibitors: 4-sulfamoyl-benzenecarboxamides and 4-chloro-3-sulfamoyl-benzenecarboxamides with strong topical antiglaucoma properties.
Bioorganic & medicinal chemistry letters 20010709
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Design and synthesis of benzoic acid derivatives as influenza neuraminidase inhibitors using structure-based drug design.
Journal of medicinal chemistry 19971205