170364-57-5 | Enzastaurin

Packsize	Purity	Availability	Price	Discounted Price
1mg	98%	in stock	$20.00	$14.00
5mg	98%	in stock	$36.00	$25.00
10mg	98%	in stock	$50.00	$35.00
50mg	98%	in stock	$123.00	$86.00
100mg	98%	in stock	$185.00	$129.00
250mg	98%	in stock	$312.00	$218.00
1g	98%	in stock	$808.00	$565.00

Description

• Catalog Number: AE81331
• Chemical Name: Enzastaurin
• CAS Number: 170364-57-5
• Molecular Formula: C32H29N5O2
• Molecular Weight: 515.605
• MDL Number: MFCD11040980
• SMILES: O=C1NC(=O)C(=C1c1cn(c2c1cccc2)C1CCN(CC1)Cc1ccccn1)c1cn(c2c1cccc2)C

Computed Properties

• Complexity: 974
• Covalently-Bonded Unit Count: 1
• Heavy Atom Count: 39
• Hydrogen Bond Acceptor Count: 4
• Hydrogen Bond Donor Count: 1
• Rotatable Bond Count: 5
• XLogP3: 3.7

Literature

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  Annals of hematology 20121001

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• A double-blind, randomized, placebo-controlled, phase 2 study of maintenance enzastaurin with 5-fluorouracil/leucovorin plus bevacizumab after first-line therapy for metastatic colorectal cancer.

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