-
Synthesis, characterization and structure optimization of a series of thiazolidinone derivatives as Entamoeba histolytica inhibitors.
European journal of medicinal chemistry 20120901
-
Discovery and modification of sulfur-containing heterocyclic pyrazoline derivatives as potential novel class of β-ketoacyl-acyl carrier protein synthase III (FabH) inhibitors.
Bioorganic & medicinal chemistry letters 20120715
-
Recent developments and biological activities of thiazolidinone derivatives: a review.
Bioorganic & medicinal chemistry 20120601
-
Synthesis and biological evaluation of a class of 5-benzylidene-2-phenyl-thiazolinones as potent 5-lipoxygenase inhibitors.
Bioorganic & medicinal chemistry 20120601
-
Molecular pharmacological profile of a novel thiazolinone-based direct and selective 5-lipoxygenase inhibitor.
British journal of pharmacology 20120401
-
Effect of structural modifications on 3-(3,5-dichlorophenyl)-2,4-thiazolidinedione-induced hepatotoxicity in Fischer 344 rats.
Journal of applied toxicology : JAT 20120201
-
Synthesis and biological evaluation of some thiazolidinones as antimicrobial agents.
European journal of medicinal chemistry 20120201
-
Prediction of promiscuous p-glycoprotein inhibition using a novel machine learning scheme.
PloS one 20120101
-
Cellulose biosynthesis inhibitors: comparative effect on bean cell cultures.
International journal of molecular sciences 20120101
-
Synthesis of s-triazine-based thiazolidinones as antimicrobial agents.
Zeitschrift fur Naturforschung. C, Journal of biosciences 20120101
-
Cellulose synthase complexes: composition and regulation.
Frontiers in plant science 20120101
-
Accelerating forward genetics for cell wall deconstruction.
Frontiers in plant science 20120101
-
Synthesis, in vitro antitubercular activity and 3D-QSAR of novel quinoxaline derivatives.
Chemical biology & drug design 20111201
-
Cell wall integrity maintenance in plants: lessons to be learned from yeast?
Plant signaling & behavior 20111101
-
2-Imino-3-(2-nitro-phen-yl)-1,3-thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20111001
-
Design, synthesis, and evaluation of thiazolidinone derivatives as antimicrobial and anti-viral agents.
Chemical biology & drug design 20110901
-
(E)-4-Phenyl-butan-2-one oxime.
Acta crystallographica. Section E, Structure reports online 20110901
-
Brassinosteroids can regulate cellulose biosynthesis by controlling the expression of CESA genes in Arabidopsis.
Journal of experimental botany 20110801
-
Synthesis and antimalarial activity of new heterocyclic hybrids based on chloroquine and thiazolidinone scaffolds.
Bioorganic & medicinal chemistry 20110801
-
Anti-infectives: can cellular screening deliver?
Current opinion in chemical biology 20110801
-
On-tissue chemical derivatization of 3-methoxysalicylamine for MALDI-imaging mass spectrometry.
Journal of mass spectrometry : JMS 20110801
-
3-Benzyl-5-benzyl-idene-2-sulfanylidene-1,3-thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20110801
-
Role of CFTR expressed by neutrophils in modulating acute lung inflammation and injury in mice.
Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20110701
-
Cell wall damage-induced lignin biosynthesis is regulated by a reactive oxygen species- and jasmonic acid-dependent process in Arabidopsis.
Plant physiology 20110701
-
5-Benzyl-idene-3-phenyl-2-phenyl-imino-1,3-thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20110701
-
Rice Brittle culm 6 encodes a dominant-negative form of CesA protein that perturbs cellulose synthesis in secondary cell walls.
Journal of experimental botany 20110301
-
Synthesis, characterization, antioxidant and antitumor evaluation of some new thiazolidine and thiazolidinone derivatives.
Archiv der Pharmazie 20110301
-
N-[5-Methyl-2-(2-nitro-phen-yl)-4-oxo-1,3-thia-zolidin-3-yl]pyridine-3-carboxamide monohydrate.
Acta crystallographica. Section E, Structure reports online 20110201
-
Synthesis, reactions and biological evaluation of some new naphtho[2,1-b]furan derivatives bearing a pyrazole nucleus.
Molecules (Basel, Switzerland) 20110105
-
In vitro evaluation of 5-arylidene-2-thioxo-4-thiazolidinones active as aldose reductase inhibitors.
Bioorganic & medicinal chemistry letters 20110101
-
Dysfunctional CFTR alters the bactericidal activity of human macrophages against Pseudomonas aeruginosa.
PloS one 20110101
-
Synthesis and antimicrobial properties of naphthylamine derivatives having a thiazolidinone moiety.
Medicina (Kaunas, Lithuania) 20110101
-
A facile synthesis and anticancer activity evaluation of spiro[thiazolidinone-isatin] conjugates.
Scientia pharmaceutica 20110101
-
Identifying HER2 inhibitors from natural products database.
PloS one 20110101
-
Understanding Plant Cellulose Synthases through a Comprehensive Investigation of the Cellulose Synthase Family Sequences.
Frontiers in plant science 20110101
-
Mapping the follicle-stimulating hormone-induced signaling networks.
Frontiers in endocrinology 20110101
-
N-(3-Octyl-4-oxo-1,3-thia-zolidin-2-yl-idene)benzamide.
Acta crystallographica. Section E, Structure reports online 20101201
-
5-(2,3,4,5,6-Penta-fluoro-phen-yl)-1,3,4-thia-diazol-2-amine.
Acta crystallographica. Section E, Structure reports online 20101101
-
Alignment between PIN1 polarity and microtubule orientation in the shoot apical meristem reveals a tight coupling between morphogenesis and auxin transport.
PLoS biology 20101001
-
Discovery of novel PTP1B inhibitors with antihyperglycemic activity.
Acta pharmacologica Sinica 20100801
-
2-(4-Fluoro-phen-yl)-3-[5-(4-nitro-phen-yl)-1,3,4-thia-diazol-2-yl]-1,3-thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20100701
-
N-(3-Butyl-4-oxo-1,3-thia-zolidin-2-yl-idene)benzamide.
Acta crystallographica. Section E, Structure reports online 20100701
-
Natural product-inspired synthesis of thiazolidine and thiazolidinone compounds and their anticancer activities.
Current pharmaceutical design 20100601
-
Anti-parasitic action and elimination of intracellular Toxoplasma gondii in the presence of novel thiosemicarbazone and its 4-thiazolidinone derivatives.
Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas 20100201
-
(E)-1-(2,4-Dinitro-phen-yl)-2-pentyl-idenehydrazine.
Acta crystallographica. Section E, Structure reports online 20100201
-
Semipreparative HPLC enantioseparation, chiroptical properties, and absolute configuration of two novel cyclooxygenase-2 inhibitors.
Chirality 20100101
-
Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugs.
Bioorganic & medicinal chemistry 20100101
-
Design, synthesis and biological evaluation of thiazolidinone derivatives as potential EGFR and HER-2 kinase inhibitors.
Bioorganic & medicinal chemistry 20100101
-
Synthesis and in vitro antimicrobial study of Schiff base and thiazolidinone of 1-cyclopropyl-6-fluoro-7-[4-(2,3-dichlorophenyl)piperazin-1-yl]-4-quinolone.
Acta poloniae pharmaceutica 20100101
-
Habituation to thaxtomin A in hybrid poplar cell suspensions provides enhanced and durable resistance to inhibitors of cellulose synthesis.
BMC plant biology 20100101
-
Synthesis and evaluation of 1,3 di-substituted schiff, mannich bases and spiro isatin derivatives.
Journal of young pharmacists : JYP 20100101
-
Studies of Antimicrobial Activities of some 4-Thiazolidinone Fused Pyrimidines, [1,5]-Benzodiazepines and their Oxygen Substituted Hydroxylamine Derivatives.
Indian journal of pharmaceutical sciences 20100101
-
Synthesis and pharmacological evaluation of novel N-alkyl/aryl substituted thiazolidinone arecoline analogues as muscarinic receptor 1 agonist in Alzheimer's dementia models.
European journal of medicinal chemistry 20091201
-
Ionic liquid mediated and promoted eco-friendly preparation of thiazolidinone and pyrimidine nucleoside-thiazolidinone hybrids and their antiparasitic activities.
Bioorganic & medicinal chemistry letters 20091115
-
Semisynthetic latrunculin B analogs: studies of actin docking support a proposed mechanism for latrunculin bioactivity.
Bioorganic & medicinal chemistry 20091101
-
2-(2-Chloro-3-quinol-yl)-3-phenyl-thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20091101
-
Synthesis, spectral and biological evaluation of some new thiazolidinones and thiazoles based on t-3-alkyl-r-2,c-6-diarylpiperidin-4-ones.
European journal of medicinal chemistry 20091001
-
Synthesis and antitumor activity of substituted triazolo[4,3-a]pyrimidin-6-sulfonamide with an incorporated thiazolidinone moiety.
Bioorganic & medicinal chemistry letters 20090801
-
Muscarinic receptor 1 agonist activity of novel N-aryl carboxamide substituted 3-morpholino arecoline derivatives in Alzheimer's presenile dementia models.
Bioorganic & medicinal chemistry 20090801
-
N-[2-(6-Methyl-4-oxo-4H-chromen-3-yl)-4-oxothia-zolidin-3-yl]furan-2-carbox-amide N,N-dimethyl-formamide solvate.
Acta crystallographica. Section E, Structure reports online 20090801
-
Microwave assisted synthesis of unsaturated jasmone heterocyclic analogues as new fragrant substances.
European journal of medicinal chemistry 20090701
-
Synthesis and antitumor activity of some new xanthotoxin derivatives.
European journal of medicinal chemistry 20090701
-
Synthesis and biological evaluation of some thiazolidinone derivatives of steroid as antibacterial agents.
European journal of medicinal chemistry 20090601
-
N'-[(2Z)-3-Allyl-4-oxo-1,3-thia-zolidin-2-yl-idene]-5-fluoro-3-phenyl-1H-indole-2-carbohydrazide.
Acta crystallographica. Section E, Structure reports online 20090501
-
5-(4-Phenoxy-phen-yl)-1,3,4-thia-diazol-2-amine.
Acta crystallographica. Section E, Structure reports online 20090501
-
2-(4-Chloro-phen-yl)-3-p-tolyl-1,3-thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20090401
-
Synthesis of 2-(5-((5-(4-chlorophenyl)furan-2-yl)methylene)-4-oxo-2-thioxothiazolidin-3-yl)acetic acid derivatives and evaluation of their cytotoxicity and induction of apoptosis in human leukemia cells.
Bioorganic & medicinal chemistry 20090315
-
Predicting anti-HIV activity of 1,3,4-thiazolidinone derivatives: 3D-QSAR approach.
European journal of medicinal chemistry 20090301
-
Tethered thiazolidinone dimers as inhibitors of the bacterial type III secretion system.
Bioorganic & medicinal chemistry letters 20090301
-
Preclinical pharmacokinetic and pharmacodynamic evaluation of thiazolidinone PG15: an anti-inflammatory candidate.
The Journal of pharmacy and pharmacology 20090301
-
Thaxtomin A affects CESA-complex density, expression of cell wall genes, cell wall composition, and causes ectopic lignification in Arabidopsis thaliana seedlings.
Journal of experimental botany 20090301
-
2-(2,4-Diphenyl-3-aza-bicyclo-[3.3.1]nonan-9-ylidenehydrazono)-1,3-thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20090301
-
Time of the day for 11beta-HSD1 inhibition plays a role in improving glucose homeostasis in DIO mice.
Diabetes, obesity & metabolism 20090201
-
Synthesis and anti-HIV studies of 2- and 3-adamantyl-substituted thiazolidin-4-ones.
European journal of medicinal chemistry 20090101
-
Toward the discovery of vaccine adjuvants: coupling in silico screening and in vitro analysis of antagonist binding to human and mouse CCR4 receptors.
PloS one 20090101
-
Antimicrobial activity of new 2,4-disubstituted thiazolidinone derivatives.
Zeitschrift fur Naturforschung. C, Journal of biosciences 20090101
-
Tributylphosphine-catalyzed cycloaddition of aziridines with carbon disulfide and isothiocyanate.
The Journal of organic chemistry 20081121
-
Synthesis and in vitro antiproliferative activity against human cancer cell lines of novel 5-(4-methyl-benzylidene)-thiazolidine-2,4-diones.
Investigational new drugs 20081001
-
A novel, cellulose synthesis inhibitory action of ancymidol impairs plant cell expansion.
Journal of experimental botany 20081001
-
Autonomic nervous system and cardiovascular system.
Indian journal of pharmacology 20081001
-
Pioglitazone treatment stimulates circulating CD34-positive cells in type 2 diabetes patients.
Diabetes research and clinical practice 20080901
-
Thiazolidinone CFTR inhibitors with improved water solubility identified by structure-activity analysis.
Bioorganic & medicinal chemistry 20080901
-
Evidence for direct CFTR inhibition by CFTR(inh)-172 based on Arg347 mutagenesis.
The Biochemical journal 20080701
-
Small-molecule CFTR inhibitors slow cyst growth in polycystic kidney disease.
Journal of the American Society of Nephrology : JASN 20080701
-
3-[5-(4-Fluoro-phen-yl)-1,3,4-thia-diazol-2-yl]-2-(4-methoxy-phen-yl)-1,3-thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20080701
-
Alpha-aminoazaheterocyclic-methylglyoxal adducts do not inhibit cystic fibrosis transmembrane conductance regulator chloride channel activity.
The Journal of pharmacology and experimental therapeutics 20080501
-
4-Thiazolidinones: a novel class of hepatitis C virus NS5B polymerase inhibitors.
Frontiers in bioscience : a journal and virtual library 20080501
-
2-(2,4-Dichloro-phen-yl)-3-[5-(4-methoxy-phen-yl)-1,3,4-thia-diazol-2-yl]-1,3-thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20080501
-
N-(3-Oxo-1-thia-4-aza-spiro-[4.5]dec-4-yl)-6-phenyl-imidazo[2,1-b][1,3]thia-zole-3-acetamide hemihydrate.
Acta crystallographica. Section E, Structure reports online 20080501
-
Differing pharmacological activities of thiazolidinone analogs at the FSH receptor.
Biochemical and biophysical research communications 20080411
-
Reactivity of fullerene epoxide: preparation of fullerene-fused thiirane, tetrahydrothiazolidin-2-one, and 1,3-dioxolane.
The Journal of organic chemistry 20080404
-
Synthesis of new imidazolyl acetic acid derivatives with anti-inflammatory and analgesic activities.
Archives of pharmacal research 20080401
-
Design, synthesis, cytoselective toxicity, structure-activity relationships, and pharmacophore of thiazolidinone derivatives targeting drug-resistant lung cancer cells.
Journal of medicinal chemistry 20080313
-
Assessment of hypolipidaemic activity of three thiazolidin-4-ones in mice given high-fat diet and fructose.
Chemico-biological interactions 20080215
-
Insight into the early steps of root hair formation revealed by the procuste1 cellulose synthase mutant of Arabidopsis thaliana.
BMC plant biology 20080101
-
Human genetics branches out in Barcelona.
Genome biology 20080101
-
Antiinflammatory, analgesic and antipyretic activity of certain thiazolidinones.
Indian journal of pharmaceutical sciences 20080101
-
Comparative molecular field analysis of benzothiazepine derivatives: mitochondrial sodium calcium exchange inhibitors as antidiabetic agents.
Indian journal of pharmaceutical sciences 20080101
-
3-(3-Chloro-4-methyl-phen-yl)-2-(4-fluoro-phen-yl)thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20080101
-
2-(2,4-Dichloro-phen-yl)-3-[5-(3,5-dimethyl-phen-yl)-1,3,4-thia-diazol-2-yl]thia-zolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20080101
-
Synthesis and Pharmacological Evaluation of Azetidin-2-ones and Thiazolidin-4-ones Encompassing Benzothiazole.
Indian journal of pharmaceutical sciences 20080101
-
Antibacterial Activity of Barringtonia acutangula against Selected Urinary Tract Pathogens.
Indian journal of pharmaceutical sciences 20080101
-
Latrunculin with a highly oxidized thiazolidinone ring: structure assignment and actin docking.
Organic letters 20071108
-
Synthesis and antimicrobial evaluation of some new thiazole, thiazolidinone and thiazoline derivatives starting from 1-chloro-3,4-dihydronaphthalene-2-carboxaldehyde.
European journal of medicinal chemistry 20070701
-
Synthesis and biological evaluation of thiazolidine-2-one 1,1-dioxide as inhibitors of Escherichia coli beta-ketoacyl-ACP-synthase III (FabH).
Bioorganic & medicinal chemistry letters 20070215
-
Latrunculin analogues with improved biological profiles by 'diverted total synthesis': preparation, evaluation, and computational analysis.
Chemistry (Weinheim an der Bergstrasse, Germany) 20070101
-
Anticancer activity of 5-benzylidene-2-phenylimino-1, 3-thiazolidin-4-one (BPT) analogs.
Medicinal chemistry (Shariqah (United Arab Emirates)) 20061101
-
Synthesis and in vitro antitumor evaluation of some indeno[1,2-c]pyrazol(in)es substituted with sulfonamide, sulfonylurea(-thiourea) pharmacophores, and some derived thiazole ring systems.
Bioorganic & medicinal chemistry 20061001
-
Synthesis and anticonvulsant activity of some potential thiazolidinonyl 2-oxo/thiobarbituric acids.
European journal of medicinal chemistry 20061001
-
Synthesis and pharmacological activity of 2-(substituted)-3-{2-[(4-phenyl-4-cyano)piperidino]ethyl}-1,3-thiazolidin-4-ones.
Chemical biology & drug design 20060601
-
Allosteric activation of the follicle-stimulating hormone (FSH) receptor by selective, nonpeptide agonists.
The Journal of biological chemistry 20060512
-
Microwave assisted synthesis of fragrant jasmone heterocyclic analogues.
European journal of medicinal chemistry 20060501
-
Diversity of Cl(-) channels.
Cellular and molecular life sciences : CMLS 20060101
-
CFTR chloride channel drug discovery--inhibitors as antidiarrheals and activators for therapy of cystic fibrosis.
Current pharmaceutical design 20060101
-
Evidence that CFTR is expressed in rat tracheal smooth muscle cells and contributes to bronchodilation.
Respiratory research 20060101
-
Structure-based discovery of inhibitors of the YycG histidine kinase: new chemical leads to combat Staphylococcus epidermidis infections.
BMC microbiology 20060101
-
Preparation of highly substituted gamma-lactam follicle stimulating hormone receptor agonists.
Bioorganic & medicinal chemistry 20051101
-
Synthesis of new 4-oxo-2-thioxo-1,2,3,4-tetrahydropyrimidine derivatives with an incorporated thiazolidinone moiety and testing their possible serine protease and cercarial elastase inhibitory effects with a possible prospective to block penetration of Schistosoma mansoni cercariae into the mice skin.
Archives of pharmacal research 20050901
-
Anti-microbial activity and film characterization of thiazolidinone derivatives of chitosan.
Macromolecular bioscience 20050624
-
Discovery of 2-arylthiazolidine-4-carboxylic acid amides as a new class of cytotoxic agents for prostate cancer.
Journal of medicinal chemistry 20050407
-
Antidiabetic and adipogenic properties in a newly synthesized thiazolidine derivative, FPFS-410.
Metabolism: clinical and experimental 20041201
-
Syntheses and evaluation of antioxidant activity of sydnonyl substituted thiazolidinone and thiazoline derivatives.
Bioorganic & medicinal chemistry 20040901
-
Effects of a new cystic fibrosis transmembrane conductance regulator inhibitor on Cl- conductance in human sweat ducts.
Experimental physiology 20040701
-
A new dimension to the biosynthetic products isolated from the sponge Negombata magnifica.
Journal of natural products 20040601
-
Agonists of the follicle stimulating hormone receptor from an encoded thiazolidinone library.
Journal of combinatorial chemistry 20040101
-
Synthesis of some thiazolyl and thiadiazolyl derivatives of 4(3H)-quinazolinone as anti-inflammatory-antimicrobial agents.
Bollettino chimico farmaceutico 20040101
-
Tetrazolo[1,5-a] quinoline derivatives as anti-inflammatory and antimicrobial agents [1].
Bollettino chimico farmaceutico 20040101
-
Synthesis and biological evaluations of sulfa derivatives bearing heterocyclic moieties.
Bollettino chimico farmaceutico 20040101
-
Synthesis and fungicidal activity of novel 4,4'-bis(2' '-aryl-5' '-methyl/unsubstituted-4' '-oxo-thiazolidin-3' '-yl) bibenzyl.
Journal of agricultural and food chemistry 20031119
-
Synthesis of some new thiazole derivatives of pharmaceutical interest.
Bollettino chimico farmaceutico 20031101
-
Synthesis and biological investigations of new thiazolidinone and oxadiazoline coumarin derivatives.
Archives of pharmacal research 20030901
-
[5-Benzyl-3-phenyl-2-(2-pyridyl-kappaN)thiazolidin-4-one-kappaS]dichloropalladium(II).
Acta crystallographica. Section C, Crystal structure communications 20021201
-
[New substituted 4-thioxothiazolidin-2-one derivatives: synthesis and structural study].
Annales pharmaceutiques francaises 20021101
-
A new synthesis of oxadiazole, thiazolidinone, N-phthalimidoamino carbonyl and arylidene derivatives with potential antimicrobial activity.
Archiv der Pharmazie 20020601
-
Synthesis of thiaazaheterocycle nucleoside analogues.
Nucleosides, nucleotides & nucleic acids 20020101
-
Two thiazolino[2,3-a]isoquinolinone S-oxides.
Acta crystallographica. Section C, Crystal structure communications 20011201
-
The reversed Kenner linker: a new safety-catch linker for the preparation of N-alkyl sulfonamides.
Organic letters 20010920
-
Thiazolidine prodrugs as protective agents against gamma-radiation-induced toxicity and mutagenesis in V79 cells.
Journal of medicinal chemistry 20010802
-
Synthesis and evaluation of the analgesic and antiinflammatory activities of O-substituted salicylamides.
Archives of pharmacal research 20010601
