-
Daily passive cycling attenuates the hyperexcitability and restores the responsiveness of the extensor monosynaptic reflex to quipazine in the chronic spinally transected rat.
Journal of neurotrauma 20140615
-
Discovery of a tetracyclic quinoxaline derivative as a potent and orally active multifunctional drug candidate for the treatment of neuropsychiatric and neurological disorders.
Journal of medicinal chemistry 20140327
-
Sensory feedback modulates quipazine-induced stepping behavior in the newborn rat.
Behavioural brain research 20120401
-
The upright posture improves plantar stepping and alters responses to serotonergic drugs in spinal rats.
The Journal of physiology 20120401
-
Synthesis, in vitro binding studies and docking of long-chain arylpiperazine nitroquipazine analogues, as potential serotonin transporter inhibitors.
European journal of medicinal chemistry 20120301
-
Differential regulation of MeCP2 phosphorylation in the CNS by dopamine and serotonin.
Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20120101
-
Mass-spectrometric studies of new 6-nitroquipazines-serotonin transporter inhibitors.
Analytical and bioanalytical chemistry 20120101
-
Motor deficits and recovery in rats with unilateral spinal cord hemisection mimic the Brown-Sequard syndrome.
Brain : a journal of neurology 20110801
-
Cholesterol and lipid phases influence the interactions between serotonin receptor agonists and lipid bilayers.
The Journal of biological chemistry 20101231
-
Why variability facilitates spinal learning.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20100811
-
Afferent inputs to mid- and lower-lumbar spinal segments are necessary for stepping in spinal cats.
Annals of the New York Academy of Sciences 20100601
-
A novel 5-HT(2A) receptor antagonist exhibits antidepressant-like effects in a battery of rodent behavioural assays: approaching early-onset antidepressants.
Pharmacology, biochemistry, and behavior 20100101
-
The interactions of the 5-HT3 receptor with quipazine-like arylpiperazine ligands: the journey track at the end of the first decade of the third millennium.
Current topics in medicinal chemistry 20100101
-
Effects of serotonergic agents on survival and hemolymph composition of the larval mosquito Aedes aegypti (Diptera: Culicidae, L.) in vivo: does serotonin regulate hemolymph acid-base homeostasis?
The Journal of experimental biology 20091101
-
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Nature chemical biology 20091001
-
Transformation of nonfunctional spinal circuits into functional states after the loss of brain input.
Nature neuroscience 20091001
-
Specific targeting of peripheral serotonin 5-HT(3) receptors. Synthesis, biological investigation, and structure-activity relationships.
Journal of medicinal chemistry 20090611
-
Synthesis and preliminary screening of novel N-{2-[4-(substituted)piperazin-1-yl]-2-oxoethyl}acetamides as potential atypical antipsychotic agents.
Journal of enzyme inhibition and medicinal chemistry 20090601
-
Serotonin receptor agonist quipazine promotes proliferation and apoptosis of human hepatocyte strain of L-02 strain.
Hepatobiliary & pancreatic diseases international : HBPD INT 20090601
-
Morphofunctional study of injured spinal cord of rats after activation of serotonergic receptors and motor load.
Doklady biological sciences : proceedings of the Academy of Sciences of the USSR, Biological sciences sections 20090101
-
Synthesis and biological evaluation of one novel technetium-99m-labeled nitroquipazine derivative as an imaging agent for serotonin transporter.
Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine 20081201
-
Synthesis and preliminary pharmacological evaluation of N-2-(4-(4-(2-substitutedthiazol-4-yl) piperazin-1-yl)-2-oxoethyl)acetamides as novel atypical antipsychotic agents.
Bioorganic & medicinal chemistry letters 20081201
-
Role of spinal 5-HT2 receptor subtypes in quipazine-induced hindlimb movements after a low-thoracic spinal cord transection.
The European journal of neuroscience 20081201
-
Dose dependence of the 5-HT agonist quipazine in facilitating spinal stepping in the rat with epidural stimulation.
Neuroscience letters 20080627
-
Epidural spinal cord stimulation plus quipazine administration enable stepping in complete spinal adult rats.
Journal of neurophysiology 20071101
-
Syntheses and binding affinities of 6-nitroquipazine analogues for serotonin transporter. Part 5: 2'-Substituted 6-nitroquipazines.
Bioorganic & medicinal chemistry 20070515
-
Presynaptic modulation of 5-HT release in the rat septal region.
Neuroscience 20070511
-
Behavioral and neuropharmacological evidence that serotonin crosses the blood-brain barrier in Coturnix japonica (Galliformes; Aves).
Brazilian journal of biology = Revista brasleira de biologia 20070201
-
[Effect of local microapplication of serotoninergic drugs on membrane currents of Paracentrotus lividus early embryos].
Ontogenez 20070101
-
Effect of robotic-assisted treadmill training and chronic quipazine treatment on hindlimb stepping in spinally transected rats.
Journal of neurotrauma 20060701
-
Presynaptic serotonergic modulation of 5-HT and acetylcholine release in the hippocampus and the cortex of 5-HT1B-receptor knockout mice.
Brain research bulletin 20060615
-
Spinal cord-transected mice learn to step in response to quipazine treatment and robotic training.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20051214
-
Preclinical pharmacology of FMPD [6-fluoro-10-[3-(2-methoxyethyl)-4-methyl-piperazin-1-yl]-2-methyl-4H-3-thia-4,9-diaza-benzo[f]azulene]: a potential novel antipsychotic with lower histamine H1 receptor affinity than olanzapine.
The Journal of pharmacology and experimental therapeutics 20051201
-
Is the platelet serotonin transporter different in venous vs. arterial blood?
Neurochemical research 20051101
-
Design and synthesis of long-chain arylpiperazines with mixed affinity for serotonin transporter (SERT) and 5-HT(1A) receptor.
The Journal of pharmacy and pharmacology 20051001
-
Effects of quipazine and m-chlorophenylbiguanide (m-CPBG) on temporal differentiation: evidence for the involvement of 5-HT2A but not 5-HT3 receptors in interval timing behaviour.
Psychopharmacology 20050901
-
Syntheses and binding affinities of 6-nitroquipazine analogues for serotonin transporter. Part 4: 3-Alkyl-4-halo-6-nitroquipazines.
Bioorganic & medicinal chemistry 20050815
-
Long-lasting recovery of locomotor function in chronic spinal rat following chronic combined pharmacological stimulation of serotonergic receptors with 8-OHDPAT and quipazine.
Neuroscience letters 20050801
-
Hyperglycemia induced by pharmacological activation of central serotonergic pathways depends on the functional integrity of brain CRH system and 5-HT3 receptors.
Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme 20050801
-
N1/P2 component of auditory evoked potential reflect changes of the brain serotonin biosynthesis in rats.
Nutritional neuroscience 20050801
-
The serotonergic agonists quipazine, CGS-12066A, and alpha-methylserotonin alter motor activity and induce hindlimb stepping in the intact and spinal rat fetus.
Behavioral neuroscience 20050601
-
Structure-affinity relationship studies on arylpiperazine derivatives related to quipazine as serotonin transporter ligands. Molecular basis of the selectivity SERT/5HT3 receptor.
Bioorganic & medicinal chemistry 20050516
-
Effects of quipazine and m-chlorophenylbiguanide (m-CPBG) on the discrimination of durations: evidence for the involvement of 5-HT2A but not 5-HT3 receptors.
Behavioural pharmacology 20050201
-
Involvement of the retinohypothalamic tract in the photic-like effects of the serotonin agonist quipazine in the rat.
Neuroscience 20050101
-
Effect of valproic acid on serotonin-2A receptor signaling in C6 glioma cells.
Journal of neurochemistry 20040901
-
Differential effects of 5-HT1 and 5-HT2 receptor agonists on hindlimb movements in paraplegic mice.
Progress in neuro-psychopharmacology & biological psychiatry 20040901
-
Synergistic activation of the central pattern generator for locomotion by l-beta-3,4-dihydroxyphenylalanine and quipazine in adult paraplegic mice.
Neuroscience letters 20040325
-
Role of NMDA receptor activation in serotonin agonist-induced air-stepping in paraplegic mice.
Spinal cord 20040301
-
Serotonin patterns locomotor network activity in the developing zebrafish by modulating quiescent periods.
Journal of neurobiology 20031201
-
Syntheses and binding affinities of 6-nitroquipazine analogues for serotonin transporter: Part 3. A potential 5-HT transporter imaging agent, 3-(3-[18F]fluoropropyl)-6-nitroquipazine.
Bioorganic & medicinal chemistry 20031117
-
5-HT1A receptors are involved in short- and long-term processes responsible for 5-HT-induced locomotor function recovery in chronic spinal rat.
The European journal of neuroscience 20031001
-
Identification of two serine residues essential for agonist-induced 5-HT2A receptor desensitization.
Biochemistry 20030916
-
Biochemical evidence for the presence of serotonin transporters in the rat cochlea.
Hearing research 20030801
-
Role of 5-HT3 receptors in the mechanisms of central pain syndrome.
Bulletin of experimental biology and medicine 20030601
-
Response of the mouse circadian system to serotonin 1A/2/7 agonists in vivo: surprisingly little.
Journal of biological rhythms 20030401
-
Thyrotropin-releasing hormone mediates serotonin-induced secretion of GH in cattle.
Domestic animal endocrinology 20030301
-
Synthesis, radiolabeling and preliminary biological evaluation of radiolabeled 5-methyl-6-nitroquipazine, a potential radioligand for the serotonin transporter.
Bioorganic & medicinal chemistry letters 20021216
-
Effects of serotonin 1A agonist on acute spinal cord injury.
Spinal cord 20021001
-
Synthesis of a fluorine-18-labelled derivative of 6-nitroquipazine, as a radioligand for the in vivo serotonin transporter imaging with PET.
Bioorganic & medicinal chemistry 20020801
-
Metachlorophenylpiperazine (m-CPP) induced intracavernous pressure responses in anaesthetized rats.
International journal of impotence research 20020801
-
Locomotor recovery in the chronic spinal rat: effects of long-term treatment with a 5-HT2 agonist.
The European journal of neuroscience 20020801
-
PET examination of [(11)C]5-methyl-6-nitroquipazine, a radioligand for visualization of the serotonin transporter.
Nuclear medicine and biology 20020801
-
Evidence for serotonergic modulation of progesterone-induced hyperphagia, depression and algesia in female mice.
Brain research 20020712
-
Electroencephalographic activation by tacrine, deprenyl, and quipazine: cholinergic vs. non-cholinergic contributions.
European journal of pharmacology 20020628
-
The Interactions of the 5-HT(3) receptor with arylpiperazine, tropane, and quinuclidine ligands.
Current topics in medicinal chemistry 20020601
-
Stimulus generalization by fenfluramine in a quipazine-ketanserin drug discrimination is not dependent on indirect serotonin release.
Pharmacology, biochemistry, and behavior 20020501
-
Serotonin sets the day state in the neurons that control coupling between the optic lobe circadian pacemakers in the cricket Gryllus bimaculatus.
The Journal of experimental biology 20020501
-
Syntheses and binding affinities of 6-nitroquipazine analogues for serotonin transporter. Part 2: 4-substituted 6-nitroquipazines.
Bioorganic & medicinal chemistry letters 20020311
-
Serotonergic attenuation of the reinforcing and neurochemical effects of cocaine in squirrel monkeys.
The Journal of pharmacology and experimental therapeutics 20020301
-
Comparison of the potency of MDL 100,907 and SB 242084 in blocking the serotonin (5-HT)(2) receptor agonist-induced increases in rat serum corticosterone concentrations: evidence for 5-HT(2A) receptor mediation of the HPA axis.
Neuropharmacology 20020201
-
Studies on modulation of feeding behavior by atypical antipsychotics in female mice.
Progress in neuro-psychopharmacology & biological psychiatry 20020201
-
RNA-editing of the 5-HT(2C) receptor alters agonist-receptor-effector coupling specificity.
British journal of pharmacology 20010901
-
Acute trazodone and quipazine treatment attenuates apomorphine-induced aggressive behaviour in male rats without major impact on emotional behaviour or monoamine content post mortem.
Pharmacological research 20010401
-
In vitro and in vivo ligand binding to the 5HT(3) serotonin receptor characterised by time-resolved fluorescence spectroscopy.
Chembiochem : a European journal of chemical biology 20010302
-
Addition of a 5-HT receptor agonist to methylphenidate potentiates the reduction of [123I]FP-CIT binding to dopamine transporters in rat frontal cortex and hippocampus.
Synapse (New York, N.Y.) 20010301
-
Neural circuits regulating pulsatile luteinizing hormone release in the female guinea-pig: opioid, adrenergic and serotonergic interactions.
Journal of neuroendocrinology 20010301
-
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 1. Mapping the central 5-HT3 receptor binding site by arylpiperazine derivatives.
Journal of medicinal chemistry 19980226
-
Similarities and differences between the subchronic and withdrawal effects of clozapine and olanzapine on forelimb force steadiness.
Psychopharmacology 19970801
-
Neurochemical and behavioral evidence that quipazine-ketanserin discrimination is mediated by serotonin2A receptor.
The Journal of pharmacology and experimental therapeutics 19951101
-
Ziprasidone (CP-88,059): a new antipsychotic with combined dopamine and serotonin receptor antagonist activity.
The Journal of pharmacology and experimental therapeutics 19951001
-
The interaction of trichloroethanol with murine recombinant 5-HT3 receptors.
British journal of pharmacology 19950401
-
REM sleep deprivation changes behavioral response to catecholaminergic and serotonergic receptor activation in rats.
Pharmacology, biochemistry, and behavior 19810701
-
Effect of drugs influencing central 5-hydroxytryptaminergic mechanisms on morphine-induced catalepsy in the rat.
The Journal of pharmacy and pharmacology 19790401
-
Effect of drugs influencing central serotonergic mechanisms on haloperidol-induced catalepsy.
Psychopharmacology 19790329
-
A combination therapy of neural and glial restricted precursor cells and chronic quipazine treatment paired with passive cycling promotes quipazine-induced stepping in adult spinalized rats.
The journal of spinal cord medicine
