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Anti-androgenic effects of S-40542, a novel non-steroidal selective androgen receptor modulator (SARM) for the treatment of benign prostatic hyperplasia.
The Prostate 20121001
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Highly regioselective synthesis of polysubstituted tetrahydroquinolines by an iodine-induced tandem cyclization reaction from propargylic alcohols and amines.
Chemistry, an Asian journal 20120901
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Oxygen and temperature sensitivity of blue to green to yellow light-emitting Pt(II) complexes.
Dalton transactions (Cambridge, England : 2003) 20120828
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Subtle structural changes in tetrahydroquinolines, a new class of nonsteroidal selective androgen receptor modulators, induce different functions.
Journal of chemical information and modeling 20120827
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An asymmetric organocatalytic Povarov reaction with 2-hydroxystyrenes.
The Journal of organic chemistry 20120817
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The asymmetric synthesis of CF3- or -CF2-substituted tetrahydroquinolines by employing a chiral phosphoric acid as catalyst.
Chemical communications (Cambridge, England) 20120811
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Synthesis of anisotropic PbS nanoparticles using heterocyclic dithiocarbamate complexes.
Dalton transactions (Cambridge, England : 2003) 20120721
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Exploration of forbidden Povarov processes as a source of unexpected reactivity: a multicomponent Mannich-Ritter transformation.
Angewandte Chemie (International ed. in English) 20120709
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Asymmetric synthesis of 2-alkyl-substituted tetrahydroquinolines by an enantioselective aza-Michael reaction.
Organic & biomolecular chemistry 20120614
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Design and synthesis of new tetrahydroquinolines derivatives as CETP inhibitors.
Bioorganic & medicinal chemistry letters 20120601
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Cyclocondensation of amino-propargyl silanes.
Organic letters 20120504
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Catalytic asymmetric synthesis of chromenes and tetrahydroquinolines via sequential allylic alkylation and intramolecular Heck coupling.
Chemical communications (Cambridge, England) 20120418
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Highly enantioselective assembly of functionalized tetrahydroquinolines with creation of an all-carbon quaternary center.
Chemistry (Weinheim an der Bergstrasse, Germany) 20120326
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1,2,3,4-tetrahydroquinoline-based selective human neuronal nitric oxide synthase (nNOS) inhibitors: lead optimization studies resulting in the identification of N-(1-(2-(methylamino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide as a preclinical development candidate.
Journal of medicinal chemistry 20120322
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Synthesis of polysubstituted, functionalized quinolines through a metal-free domino process involving a C4–C3 functional group rearrangement.
Organic letters 20120316
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2D Chemometrics analyses of tetrahydroquinoline and ethylenediamine derivatives with antimalarial activity.
Medicinal chemistry (Shariqah (United Arab Emirates)) 20120301
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Step-economical synthesis of tetrahydroquinolines by asymmetric relay catalytic Friedländer condensation/transfer hydrogenation.
Angewandte Chemie (International ed. in English) 20120116
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Ocular pharmacokinetics of a novel tetrahydroquinoline analog in rabbit: compartmental analysis and PK-PD evaluation.
Journal of pharmaceutical sciences 20120101
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The novel non-steroidal selective androgen receptor modulator S-101479 has additive effects with bisphosphonate, selective estrogen receptor modulator, and parathyroid hormone on the bones of osteoporotic female rats.
Biological & pharmaceutical bulletin 20120101
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Ocular hypotensive action of a novel tetrahydroquinoline analog in rabbit: physicochemical evaluation.
Journal of pharmaceutical sciences 20111201
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Ocular pharmacokinetics of a novel tetrahydroquinoline analog in rabbit: absorption, disposition, and non-compartmental analysis.
Journal of pharmaceutical sciences 20111201
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Cardiomyocyte death: mechanisms and translational implications.
Cell death & disease 20111201
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Advances in the chemistry of tetrahydroquinolines.
Chemical reviews 20111109
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Tetrahydroquinolines as a novel series of nonsteroidal selective androgen receptor modulators: structural requirements for better physicochemical and biological properties.
Bioorganic & medicinal chemistry letters 20111101
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Efficient synthesis and free-radical scavenging capacity of new 2,4-substituted tetrahydroquinolines prepared via BiCl₃-catalyzed three-component Povarov reaction, using N-vinylamides.
Molecular diversity 20111101
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2-Oxo-N-aryl-1,2,3,4-tetrahydroquinoline-6-sulfonamides as activators of the tumor cell specific M2 isoform of pyruvate kinase.
Bioorganic & medicinal chemistry letters 20111101
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Chiral phosphoric acid-catalyzed enantioselective three-component Povarov reaction using enecarbamates as dienophiles: highly diastereo- and enantioselective synthesis of substituted 4-aminotetrahydroquinolines.
Journal of the American Chemical Society 20110921
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Photobehavior of mixed nπ*/ππ* triplets: simultaneous detection of the two transients, solvent-dependent hydrogen abstraction, and reequilibration upon protein binding.
The journal of physical chemistry. B 20110915
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Acta crystallographica. Section E, Structure reports online 20110901
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Ring opening/C-N cyclization of activated aziridines with carbon nucleophiles: highly diastereo- and enantioselective synthesis of tetrahydroquinolines.
Organic letters 20110819
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Design, synthesis, and biological evaluation of 3,4-dihydroquinolin-2(1H)-one and 1,2,3,4-tetrahydroquinoline-based selective human neuronal nitric oxide synthase (nNOS) inhibitors.
Journal of medicinal chemistry 20110811
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Discovery, structure-activity relationship studies, and crystal structure of nonpeptide inhibitors bound to the Shank3 PDZ domain.
ChemMedChem 20110801
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FeCl3-mediated synthesis of polysubstituted tetrahydroquinolines via domino Mannich/Friedel-Crafts reactions of aldehydes and amines.
Organic & biomolecular chemistry 20110721
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Multicomponent assembly and diversification of novel heterocyclic scaffolds derived from 2-arylpiperidines.
Organic letters 20110617
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Conjugate addition of lithium N-phenyl-N-(α-methylbenzyl)amide: application to the asymmetric synthesis of (R)-(-)-angustureine.
Organic letters 20110520
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Selective activation of enantiotopic C(sp3)-hydrogen by means of chiral phosphoric acid: asymmetric synthesis of tetrahydroquinoline derivatives.
Journal of the American Chemical Society 20110427
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Dyeing behaviours of amino heterocyclic compounds as blue oxidative hair dye precursors applied to keratin fibres.
International journal of cosmetic science 20110401
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Discovery of orally available tetrahydroquinoline-based glucocorticoid receptor agonists.
Bioorganic & medicinal chemistry letters 20110315
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Design and synthesis of tricyclic tetrahydroquinolines as a new series of nonsteroidal selective androgen receptor modulators (SARMs).
Bioorganic & medicinal chemistry letters 20110315
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Tetrahydroquinolin-3-yl carbamate glucocorticoid receptor agonists with reduced PEPCK activation.
Bioorganic & medicinal chemistry letters 20110315
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A theoretical study of the mechanism for the homogeneous catalytic reversible dehydrogenation-hydrogenation of nitrogen heterocycles.
Physical chemistry chemical physics : PCCP 20110307
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Highly enantioselective synthesis of polysubstituted tetrahydroquinolines via organocatalytic Michael/Aza-Henry tandem reactions.
Organic letters 20110304
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Chroman and tetrahydroquinoline ureas as potent TRPV1 antagonists.
Bioorganic & medicinal chemistry letters 20110301
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Highly enantioselective synthesis of tetrahydroquinolines via cobalt(II)-catalyzed tandem 1,5-hydride transfer/cyclization.
Organic letters 20110218
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Scandium(III) zeolites as new heterogeneous catalysts: [4+2]cyclocondensation of in situ generated aryl imines with alkenes.
Chemistry (Weinheim an der Bergstrasse, Germany) 20110207
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Cytotoxic effects of new trans-2,4-diaryl-r-3-methyl-1,2,3,4-tetrahydroquinolines and their interaction with antitumoral drugs gemcitabine and paclitaxel on cellular lines of human breast cancer.
Chemico-biological interactions 20110201
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Cannabinoid CB(1) receptor ligand binding and function examined through mutagenesis studies of F200 and S383.
European journal of pharmacology 20110125
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Tetrahydroquinoline derivatives as opioid receptor antagonists.
Bioorganic & medicinal chemistry letters 20110115
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Natural product inspired diversity oriented synthesis of tetrahydroquinoline scaffolds as antitubercular agent.
ACS combinatorial science 20110110
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Discovery of 1-(3,4-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydroquinolin-4-amine, a dual serotonin and dopamine reuptake inhibitor.
Bioorganic & medicinal chemistry letters 20110101
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Tetrahydroquinoline glucocorticoid receptor agonists: discovery of a 3-hydroxyl for improving receptor selectivity.
Bioorganic & medicinal chemistry letters 20110101
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(3S)-2-Benzyl-3-carb-oxy-1,2,3,4-tetra-hydro-isoquinolinium chloride monohydrate.
Acta crystallographica. Section E, Structure reports online 20110101
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Non-conjugated small molecule FRET for differentiating monomers from higher molecular weight amyloid beta species.
PloS one 20110101
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Conformationally constrained histidines in the design of peptidomimetics: strategies for the χ-space control.
International journal of molecular sciences 20110101
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An essential farnesylated kinesin in Trypanosoma brucei.
PloS one 20110101
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Synthesis and Antimicrobial Activities of Some New Azetidin-2-ones and Thiazolidin-4-ones.
Indian journal of pharmaceutical sciences 20110101
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Functional importance of tyrosine 294 and the catalytic selectivity for the bis-Fe(IV) state of MauG revealed by replacement of this axial heme ligand with histidine .
Biochemistry 20101116
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Preparation of half-metallocenes of thiophene-fused and tetrahydroquinoline-linked cyclopentadienyl ligands for ethylene/α-olefin copolymerization.
Dalton transactions (Cambridge, England : 2003) 20101107
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InCl3-catalyzed allylic Friedel-Crafts reactions toward the stereocontrolled synthesis of 1,2,3,4-tetrahydroquinolines.
Organic letters 20101105
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Comparison of the activity of non-steroidal ecdysone agonists between dipteran and lepidopteran insects, using cell-based EcR reporter assays.
Pest management science 20101101
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Synthesis, testing and structure-activity studies on a library of 5-HT₄ ligands.
Medicinal chemistry (Shariqah (United Arab Emirates)) 20101101
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Quinoline-based compounds as modulators of HIV transcription through NF-kappaB and Sp1 inhibition.
Antiviral research 20100901
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Enantioselective organocatalytic C-H bond functionalization via tandem 1,5-hydride transfer/ring closure: asymmetric synthesis of tetrahydroquinolines.
Journal of the American Chemical Society 20100901
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5,8-Dimeth-oxy-2-phenyl-1,4-dihydro-quinoline-3-carbonitrile.
Acta crystallographica. Section E, Structure reports online 20100901
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A small-molecule oxocarbazate inhibitor of human cathepsin L blocks severe acute respiratory syndrome and ebola pseudotype virus infection into human embryonic kidney 293T cells.
Molecular pharmacology 20100801
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Quinaphos and Dihydro-Quinaphos phosphine-phosphoramidite ligands for asymmetric hydrogenation.
Chemistry (Weinheim an der Bergstrasse, Germany) 20100705
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Palladium-catalyzed ring-expansion reaction of indoles with alkynes: from indoles to tetrahydroquinoline derivatives under mild reaction conditions.
Angewandte Chemie (International ed. in English) 20100601
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Asymmetric three-component inverse electron-demand aza-Diels-Alder reaction: efficient synthesis of ring-fused tetrahydroquinolines.
Angewandte Chemie (International ed. in English) 20100517
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Highly efficient synthesis and characterization of the GPR30-selective agonist G-1 and related tetrahydroquinoline analogs.
Organic & biomolecular chemistry 20100507
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Assessment of species specificity of moulting accelerating compounds in Lepidoptera: comparison of activity between Bombyx mori and Spodoptera littoralis by in vitro reporter and in vivo toxicity assays.
Pest management science 20100501
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Discovering some novel tetrahydroquinoline derivatives bearing the biologically active sulfonamide moiety as a new class of antitumor agents.
European journal of medicinal chemistry 20100501
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Diverse effects on mitochondrial and nuclear functions elicited by drugs and genetic knockdowns in bloodstream stage Trypanosoma brucei.
PLoS neglected tropical diseases 20100501
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Iridium-catalyzed, silyl-directed borylation of nitrogen-containing heterocycles.
Journal of the American Chemical Society 20100331
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Diphosphine-catalyzed mixed double-Michael reaction: a unified synthesis of indolines, dihydropyrrolopyridines, benzimidazolines, tetrahydroquinolines, tetrahydroisoquinolines, dihydrobenzo-1,4-oxazines, and dihydrobenzo-3,1-oxazines.
Organic letters 20100305
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Novel tetrahydrochinoline derived CETP inhibitors.
Bioorganic & medicinal chemistry letters 20100301
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Zn(OTf)2-catalyzed reactions of ethenetricarboxylates with 2-aminobenzaldehydes leading to tetrahydroquinoline derivatives.
The Journal of organic chemistry 20100219
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Efficient entry into 2-substituted tetrahydroquinoline systems through alkylative ring expansion: stereoselective formal synthesis of (+/-)-martinellic acid.
The Journal of organic chemistry 20100205
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Easy access to isoquinolines and tetrahydroquinolines from ketoximes and alkynes via rhodium-catalyzed C-H bond activation.
The Journal of organic chemistry 20091218
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Tetrahydroquinoline derivatives as CRTH2 antagonists.
Bioorganic & medicinal chemistry letters 20091215
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N,1-Bis(4-chloro-2-methyl-benz-yl)-3-methyl-2-oxo-1,2,3,4-tetra-hydro-quinoline-3-carboxamide.
Acta crystallographica. Section E, Structure reports online 20091201
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Tetrahydroquinoline sulfonamides as vasopressin 1b receptor antagonists.
Bioorganic & medicinal chemistry letters 20091101
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Design, synthesis and anticancer evaluation of novel tetrahydroquinoline derivatives containing sulfonamide moiety.
European journal of medicinal chemistry 20091001
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Substituted tetrahydroquinolines as potent allosteric inhibitors of reverse transcriptase and its key mutants.
Bioorganic & medicinal chemistry letters 20090901
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Gold-catalyzed intramolecular allylic amination of 2-tosylaminophenylprop-1-en-3-ols. A concise synthesis of (+/-)-angustureine.
The Journal of organic chemistry 20090821
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Design and synthesis of indole, 2,3-dihydro-indole, and 3,4-dihydro-2H-quinoline-1-carbothioic acid amide derivatives as novel HCV inhibitors.
Bioorganic & medicinal chemistry letters 20090801
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Improved asymmetric synthesis of 3,4-dihydro-2-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]-5-[3-(trifluoromethoxy)phenyl]-alpha-(trifluoromethyl)-1(2H)-quinolineethanol, a potent cholesteryl ester transfer protein inhibitor.
Organic letters 20090702
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Design and synthesis of potent inhibitors of cholesteryl ester transfer protein (CETP) exploiting a 1,2,3,4-tetrahydroquinoline platform.
Bioorganic & medicinal chemistry letters 20090501
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Self-assembly of hydrogensquarates: crystal structures and properties.
The journal of physical chemistry. A 20090402
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Substituted 1,2,3,4-tetrahydroquinolin-6-yloxypropanes as beta3-adrenergic receptor agonists: design, synthesis, biological evaluation and pharmacophore modeling.
Bioorganic & medicinal chemistry 20090115
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Lewis acid or Brønsted acid catalyzed reactions of vinylidene cyclopropanes with activated carbon-nitrogen, nitrogen-nitrogen, and iodine-nitrogen double-bond-containing compounds.
Chemistry (Weinheim an der Bergstrasse, Germany) 20090101
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Synthesis and biotransformation of tetrahydroquinoline by Mortierella isabelina.
Zeitschrift fur Naturforschung. C, Journal of biosciences 20090101
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QSAR study on tetrahydroquinoline analogues as plasmodium protein farnesyltransferase inhibitors: a comparison of rationales of malarial and mammalian enzyme inhibitory activities for selectivity.
European journal of medicinal chemistry 20081201
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Air-stable and phosphine-free iridium catalysts for highly enantioselective hydrogenation of quinoline derivatives.
Organic letters 20081120
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Bis(1,2,3,4-tetra-hydro-quinolin-6-yl)methane.
Acta crystallographica. Section E, Structure reports online 20080901
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Ruthenium-catalyzed enantioselective carbon-carbon bond forming reaction via allenylidene-ene process: synthetic approach to chiral heterocycles such as chromane, thiochromane, and 1,2,3,4-tetrahydroquinoline derivatives.
Journal of the American Chemical Society 20080813
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Natural products as an inspiration in the diversity-oriented synthesis of bioactive compound libraries.
Natural product reports 20080801
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Synthesis and characterization of 5,6,7,8-tetrahydroquinoline C5a receptor antagonists.
Bioorganic & medicinal chemistry letters 20080415
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Suzuki-Miyaura approach to JNJ-26076713, an orally active tetrahydroquinoline-containing alphaVbeta3/alphaVbeta5 integrin antagonist. enantioselective synthesis and stereochemical studies.
The Journal of organic chemistry 20080321
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Strictosidine synthase: mechanism of a Pictet-Spengler catalyzing enzyme.
Journal of the American Chemical Society 20080116
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Gold-catalyzed synthesis of chroman, dihydrobenzofuran, dihydroindole, and tetrahydroquinoline derivatives.
Chemistry (Weinheim an der Bergstrasse, Germany) 20080101
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Selective androgen receptor modulators in preclinical and clinical development.
Nuclear receptor signaling 20080101
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Development of pinene-derived N,P ligands and their utility in catalytic asymmetric hydrogenation.
Dalton transactions (Cambridge, England : 2003) 20071221
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Effect of ecdysone receptor gene switch ligands on endogenous gene expression in 293 cells.
The FEBS journal 20071101
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Design, synthesis, and evaluation of tetrahydroquinoline and pyrrolidine sulfonamide carbamates as gamma-secretase inhibitors.
Bioorganic & medicinal chemistry letters 20070601
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Cobaltpolyoxometalate-catalyzed cyclization of glucal with aryl amines: Synthesis of 2,4-disubstituted tetrahydroquinolines.
Bioorganic & medicinal chemistry letters 20070515
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Lewis acid catalyzed reaction of arylvinylidenecyclopropanes with ethyl (arylimino)acetates: a facile synthetic protocol for pyrrolidine and 1,2,3,4-tetrahydroquinoline derivatives.
Organic letters 20070426
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Resistance mutations at the lipid substrate binding site of Plasmodium falciparum protein farnesyltransferase.
Molecular and biochemical parasitology 20070301
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Chiral tetrahydroquinoline derivatives as potent anti-hyperalgesic agents in animal models of sustained inflammation and chronic neuropathic pain.
Bioorganic & medicinal chemistry letters 20070301
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Moexipril and left ventricular hypertrophy.
Vascular health and risk management 20070201
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Tetrahydroquinoline sulfonamides as gamma-secretase inhibitors.
Bioorganic & medicinal chemistry letters 20070101
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Heteroarotinoids with anti-cancer activity against ovarian cancer cells.
The open medicinal chemistry journal 20070101
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Metabolic aromatization of N-alkyl-1,2,3,4-tetrahydroquinoline substructures to quinolinium by human liver microsomes and horseradish peroxidase.
Drug metabolism and disposition: the biological fate of chemicals 20061201
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Microwave-assisted, solid-phase synthesis of a chiral 1,2,3,4-tetrahydro-quinoline library.
Combinatorial chemistry & high throughput screening 20061101
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Chiral Brønsted acid-catalyzed inverse electron-demand aza Diels-Alder reaction.
Journal of the American Chemical Society 20061011
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Synthesis and stereochemical investigations of novel nitrogen-containing 13alpha-estrone derivatives.
Steroids 20060701
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Synthesis and SAR of novel histamine H3 receptor antagonists.
Bioorganic & medicinal chemistry letters 20060701
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Homoleptic rare earth dipyridylamides [Ln2(N(NC5H4)2)6], Ln = Ce, Nd, Sm, Ho, Er, Tm, Yb, and Sc: metal oxidation by the amine melt and in 1,2,3,4-tetrahydroquinoline with the focus of different metal activation by amalgams, liquid ammonia, and microwaves.
Inorganic chemistry 20060320
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Structure-activity relationships of a series of tariquidar analogs as multidrug resistance modulators.
Bioorganic & medicinal chemistry 20060301
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Adding pharmacogenomics to the development of new marine-derived anticancer agents.
Journal of translational medicine 20060101
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Synthesis, spectral studies and in vitro assessment for antiamoebic activity of new cyclooctadiene ruthenium(II) complexes with 5-nitrothiophene-2-carboxaldehyde thiosemicarbazones.
Bioorganic & medicinal chemistry letters 20051215
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First QSAR report on FSH receptor antagonistic activity: quantitative investigations on physico-chemical and structural features among 6-amino-4-phenyltetrahydroquinoline derivatives.
Bioorganic & medicinal chemistry letters 20051015
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Identification of photoproducts of hexahydroquinoline derivatives by GC-EI-MS and HPLC-ESI-MS.
Drug development and industrial pharmacy 20051001
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Protein farnesyltransferase inhibitors exhibit potent antimalarial activity.
Journal of medicinal chemistry 20050602
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Resistance to a protein farnesyltransferase inhibitor in Plasmodium falciparum.
The Journal of biological chemistry 20050408
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Asymmetric synthesis of novel tetrahydroquinoline derivatives with a sugar building block and their bioactivities.
Bioorganic & medicinal chemistry letters 20050401
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Structure-property relationship in py-hexahydrocinchonidine diastereomers: ab initio and NMR study.
The journal of physical chemistry. A 20050210
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Synthesis of novel steroid-tetrahydroquinoline hybrid molecules and D-homosteroids by intramolecular cyclization reactions.
Steroids 20040501
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Intramolecular arylation reactions of alkenes: a flexible approach to chromans and tetrahydroquinoline derivatives.
Journal of the American Chemical Society 20040324
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A solid-phase, library synthesis of natural-product-like derivatives from an enantiomerically pure tetrahydroquinoline scaffold.
Journal of combinatorial chemistry 20040101
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Helquinoline, a new tetrahydroquinoline antibiotic from Janibacter limosus Hel 1+.
The Journal of antibiotics 20040101
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A solution- and solid-phase approach to tetrahydroquinoline-derived polycyclics having a 10-membered ring.
Journal of combinatorial chemistry 20040101
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Solution- and solid-phase synthesis of natural product-like tetrahydroquinoline-based polycyclics having a medium size ring.
Journal of combinatorial chemistry 20040101
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The effect of remote chirality on the antibacterial activity of indolinyl, tetrahydroquinolyl and dihydrobenzoxazinyl oxazolidinones.
Bioorganic & medicinal chemistry letters 20031201
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Enantiomerically pure tetrahydroquinoline derivatives as in vivo potent antagonists of the glycine binding site associated to the NMDA receptor.
Bioorganic & medicinal chemistry letters 20031103
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1,4-benzothiazine analogues and apoptosis: structure-activity relationship.
Bioorganic & medicinal chemistry 20030731
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Synthesis and SAR of cis-1-benzoyl-1,2,3,4-tetrahydroquinoline ligands for control of gene expression in ecdysone responsive systems.
Bioorganic & medicinal chemistry letters 20030602
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Dihydropyridine-based multicomponent reactions. Efficient entry into new tetrahydroquinoline systems through Lewis acid-catalyzed formal [4 + 2] cycloadditions.
Organic letters 20030306
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Dihydropyridines in MCRs. Tandem processes leading to modular tetrahydroquinoline systems with up to 6 diversity elements.
Molecular diversity 20030101
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Ketene dithioacetals in the aza-Diels-Alder reaction with N-arylimines: a versatile approach to tetrahydroquinolines, 2,3-dihydro-4-quinolones, and 4-quinolones.
Organic letters 20021212
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Stereoselectivity in reactions of amino acids catalyzed by pyridoxal derivatives carrying rigidly-attached chirally-mounted basic groups--transamination, racemization, decarboxylation, retro-aldol reaction, and aldol condensation.
Bioorganic & medicinal chemistry 20021201
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Novel stereocontrolled addition of allylmetal reagents to alpha-imino esters: efficient synthesis of chiral tetrahydroquinoline derivatives.
The Journal of organic chemistry 20021018
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Novel, non-acylguanidine-type Na(+)/H(+) exchanger inhibitors: synthesis and pharmacology of 5-tetrahydroquinolinylidene aminoguanidine derivatives.
Journal of medicinal chemistry 20020704
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InCl(3)-catalyzed domino reaction of aromatic amines with cyclic enol ethers in water: a highly efficient synthesis of new 1,2,3,4-tetrahydroquinoline derivatives.
The Journal of organic chemistry 20020531
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Syntheses of fused heterocyclic compounds and their inhibitory activities for squalene synthase.
Bioorganic & medicinal chemistry 20020201
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Antiplasmodial and cytotoxic activity of galipinine and other tetrahydroquinolines from Galipea officinalis.
Planta medica 20020101
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Indole synthesis by radical cyclization of o-alkenylphenyl isocyanides and its application to the total synthesis of natural products.
Chemical record (New York, N.Y.) 20020101
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Combinatorial synthetic design. Solution and polymer-supported synthesis of heterocycles via intramolecular aza Diels-Alder and imino alcohol cyclizations.
Journal of combinatorial chemistry 20020101
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First asymmetric synthesis of quinoline derivatives by inverse electron demand (IED) Diels-Alder reaction using chiral Ti(IV) complex.
Organic letters 20010628
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Asymmetric synthesis of functionalized 1,2,3,4-tetrahydroquinolines.
Organic letters 20010628
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Diastereoselective synthesis of substituted tetrahydroquinoline-4-carboxylic esters by a tandem reduction-reductive amination reaction.
The Journal of organic chemistry 20010420
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Synthesis of a novel series of cytotoxic bisindole alkaloids.
Bioorganic & medicinal chemistry letters 20010108
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Polymer-supported glyoxylate and alpha-imino acetates. Versatile reagents for the synthesis of alpha-hydroxycarboxylic acid and alpha-amino acid libraries.
Journal of combinatorial chemistry 20010101
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Polymer-supported benzotriazoles as catalysts in the synthesis of tetrahydroquinolines by condensation of aldehydes with aromatic amines.
Journal of combinatorial chemistry 20010101
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Identification of the alkaloids of Galipea officinalis by gas chromatography-mass spectrometry.
Phytochemical analysis : PCA 20010101