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M2 muscarinic acetylcholine receptors regulate long-term potentiation at hippocampal CA3 pyramidal cell synapses in an input-specific fashion.
Journal of neurophysiology 20120701
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Translating clinical findings into knowledge in drug safety evaluation--drug induced liver injury prediction system (DILIps).
PLoS computational biology 20111201
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Role of TNF-α in virus-induced airway hyperresponsiveness and neuronal M₂ muscarinic receptor dysfunction.
British journal of pharmacology 20110901
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[Intravenous procaine as analgesic in obstetrics. 1955].
Ginecologia y obstetricia de Mexico 20110201
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Changes in blood pressure induced by electrical stimulation of the femur in anesthetized rats.
Autonomic neuroscience : basic & clinical 20101208
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A predictive ligand-based Bayesian model for human drug-induced liver injury.
Drug metabolism and disposition: the biological fate of chemicals 20101201
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Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.
Bioorganic & medicinal chemistry letters 20101101
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[Three auxiliary medications in obstetrics. 1955].
Ginecologia y obstetricia de Mexico 20101101
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A fluorescence anisotropy assay for the muscarinic M1 G-protein-coupled receptor.
Assay and drug development technologies 20100601
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Investigating the interaction of McN-A-343 with the M2 muscarinic receptor using its nitrogen mustard derivative.
Biochemical pharmacology 20100401
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A fluorescence resonance energy transfer-based M2 muscarinic receptor sensor reveals rapid kinetics of allosteric modulation.
The Journal of biological chemistry 20100319
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The effect of memantine and levodopa/carbidopa on the responses of phrenic nerve-diaphragm preparations from aged rats.
Medical science monitor : international medical journal of experimental and clinical research 20091101
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Kinetics of inhibition of acetylcholinesterase in the presence of acetonitrile.
The FEBS journal 20090401
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An in vitro model for studying neuromuscular transmission in the mouse pharynx.
Dysphagia 20090301
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Use of acetylcholine mustard to study allosteric interactions at the M(2) muscarinic receptor.
The Journal of pharmacology and experimental therapeutics 20081101
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Acute anal stretch inhibits NMDA-dependent pelvic-urethra reflex potentiation via spinal GABAergic inhibition in anesthetized rats.
American journal of physiology. Renal physiology 20081001
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Binding of orthosteric ligands to the allosteric site of the M(2) muscarinic cholinergic receptor.
Molecular pharmacology 20080901
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Two-state models and the analysis of the allosteric effect of gallamine at the M2 muscarinic receptor.
The Journal of pharmacology and experimental therapeutics 20080601
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The impact of orthosteric radioligand depletion on the quantification of allosteric modulator interactions.
The Journal of pharmacology and experimental therapeutics 20080601
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[Neuromuscular monitoring: methods and machines].
Anasthesiologie, Intensivmedizin, Notfallmedizin, Schmerztherapie : AINS 20080501
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Acetylcholine mediates the release of IL-8 in human bronchial epithelial cells by a NFkB/ERK-dependent mechanism.
European journal of pharmacology 20080317
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Subtype-selective blockade of cardiac muscarinic receptors inhibits vagal chronotropic responses in cats.
Pflugers Archiv : European journal of physiology 20080201
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Autoantibodies enhance agonist action and binding to cardiac muscarinic receptors in chronic Chagas' disease.
Journal of receptor and signal transduction research 20080101
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First gallamine-tacrine hybrid: design and characterization at cholinesterases and the M2 muscarinic receptor.
Journal of medicinal chemistry 20071115
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The effect of some curarizing drugs in unanaesthetized man. I. d-Tubocurarine chloride, gallamonium iodide, decamethonium iodide, succinylcholine iodide and its bis-monoethyl-substituted derivative in single or repeated doses. Acta Anaesth. Scandinav. 1957, 1, 15-39.
Acta anaesthesiologica Scandinavica 20070901
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Allosteric interaction of the neuromuscular blockers vecuronium and pancuronium with recombinant human muscarinic M2 receptors.
European journal of pharmacology 20070813
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Mutational disruption of a conserved disulfide bond in muscarinic acetylcholine receptors attenuates positive homotropic cooperativity between multiple allosteric sites and has subtype-dependent effects on the affinities of muscarinic allosteric ligands.
Molecular pharmacology 20070301
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Allosteric interactions with muscarinic acetylcholine receptors: complex role of the conserved tryptophan M2422Trp in a critical cluster of amino acids for baseline affinity, subtype selectivity, and cooperativity.
Molecular pharmacology 20060701
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Pharmacology and surface electrostatics of the K channel outer pore vestibule.
The Journal of membrane biology 20060701
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Inhibitory M2 muscarinic receptors are upregulated in both axotomized and intact small diameter dorsal root ganglion cells after peripheral nerve injury.
Neuroscience 20060619
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Cardiac activity and blood pressure in rats during selective blockade of various subtypes of muscarinic cholinoceptors.
Bulletin of experimental biology and medicine 20060601
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Identification of various allosteric interaction sites on M1 muscarinic receptor using 125I-Met35-oxidized muscarinic toxin 7.
Molecular pharmacology 20060501
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Effects of muscarinic antagonists on ZENK expression in the chicken retina.
Experimental eye research 20060301
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Allosteric site in M2 acetylcholine receptors: evidence for a major conformational change upon binding of an orthosteric agonist instead of an antagonist.
Naunyn-Schmiedeberg's archives of pharmacology 20060101
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Methoctramine and gallamine inhibit PI hydrolysis in guinea-pig gallbladder.
Vascular pharmacology 20051001
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Prevention of succinylcholine-induced fasciculation and myalgia: a meta-analysis of randomized trials.
Anesthesiology 20051001
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The first synthetic nondepolarizing muscle relaxant--gallamine.
Anaesthesia and intensive care 20051001
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Critical amino acid residues of the common allosteric site on the M2 muscarinic acetylcholine receptor: more similarities than differences between the structurally divergent agents gallamine and bis(ammonio)alkane-type hexamethylene-bis-[dimethyl-(3-phthalimidopropyl)ammonium]dibromide.
Molecular pharmacology 20050901
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Effects on heart rate of an anti-M2 acetylcholine receptor immune response in mice.
FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20050601
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Regulation of M2 muscarinic acetylcholine receptor expression and signaling by prolonged exposure to allosteric modulators.
The Journal of pharmacology and experimental therapeutics 20050101
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M2 muscarinic acetylcholine receptor knock-out mice show deficits in behavioral flexibility, working memory, and hippocampal plasticity.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20041110
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Effect of some cardiac and respiratory drugs on succinate-cytochrome c reductase.
Journal of enzyme inhibition and medicinal chemistry 20040801
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Two distinct classes of muscarinic action on hippocampal inhibitory synapses: M2-mediated direct suppression and M1/M3-mediated indirect suppression through endocannabinoid signalling.
The European journal of neuroscience 20040501
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Cholinergic modulation of nociceptive responses in vivo and neuropeptide release in vitro at the level of the primary sensory neuron.
Pain 20040101
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G-protein coupled receptors as allosteric machines.
Receptors & channels 20040101
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Future therapeutic strategies in autoimmune myasthenia gravis.
Annals of the New York Academy of Sciences 20030901
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Postsynaptic M1 and M3 receptors are responsible for the muscarinic enhancement of retrograde endocannabinoid signalling in the hippocampus.
The European journal of neuroscience 20030701
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An unusual form of the association binding kinetics of N-[3H]methylscopolamine to the split muscarinic M2trunk/M2tail receptor.
The Journal of pharmacology and experimental therapeutics 20030501
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Gallamine-tetraphenylborate-modified carbon paste electrode for the potentiometric determination of gallamine triethiodide (flaxedil).
Journal of pharmaceutical and biomedical analysis 20030326
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Chemically modified carbon paste electrode for iodide determination on the basis of cetyltrimethylammonium iodide ion-pair.
Analytical sciences : the international journal of the Japan Society for Analytical Chemistry 20030201
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Involvement of cholinoceptors in cadmium-induced endothelial dysfunction.
Journal of basic and clinical physiology and pharmacology 20030101
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Nuclear factor kappaB activation by muscarinic receptors in astroglial cells: effect of ethanol.
Neuroscience 20030101
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Cardiovascular effects of intravenous pentazocine and cyclazocine in conscious, curarized-conscious, and anesthetized dogs.
Journal of basic and clinical physiology and pharmacology 20030101
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Analogs of WIN 62,577 define a second allosteric site on muscarinic receptors.
Molecular pharmacology 20021201
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Role of muscarinic acetylcholine receptors in a guinea pig model of asthma.
International immunopharmacology 20021001
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The nature of the acetylcholine and 5-hydroxytryptamine receptors in buccal smooth muscle of the pest slug Deroceras reticulatum.
Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology 20020401
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Anionic cyclophanes as potential reversal agents of muscle relaxants by chemical chelation.
Bioorganic & medicinal chemistry letters 20020311
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Isobolographic analysis of non-depolarising muscle relaxant interactions at their receptor site.
European journal of pharmacology 20020301
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Muscle distribution of the neuromuscular blocker gallamine using microdialysis.
Journal of pharmaceutical sciences 20020301
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Pharmacology and chemistry of the venoms of solitary wasps.
Journal of natural toxins 20020201
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Cholinergic and serotonergic activities are required in triggering conditioned NK cell response.
Journal of neuroimmunology 20020201
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Systemic anaphylaxis induced by intradermal testing.
Allergie et immunologie 20020201
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Changes of cooperativity between N-methylscopolamine and allosteric modulators alcuronium and gallamine induced by mutations of external loops of muscarinic M(3) receptors.
Molecular pharmacology 20011001
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Muscarinic activation of inwardly rectifying K(+) conductance reduces EPSPs in rat hippocampal CA1 pyramidal cells.
The Journal of physiology 20010901
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Muscarinic allosteric modulation: M2/M3 subtype selectivity of gallamine is independent of G-protein coupling specificity.
Naunyn-Schmiedeberg's archives of pharmacology 20010801
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The influence of surface charges on quaternary ammonium block of shaker K+ channels.
The Journal of membrane biology 20010801
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Succinylcholine pretreatment using gallamine or mivacurium during rapid sequence induction in children: a randomized, controlled study.
Journal of clinical anesthesia 20010601
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Application of a high-performance liquid chromatographic assay for the neuromuscular blocker gallamine to analysis of rat plasma, muscle and microdialysate samples.
Journal of chromatography. B, Biomedical sciences and applications 20010425
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Cathodic adsorptive stripping voltammetric determination of muscle relaxant: gallamine triethiodide (flaxedil).
Journal of pharmaceutical and biomedical analysis 20010401
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Glucocorticoid treatment increases inhibitory m(2) muscarinic receptor expression and function in the airways.
American journal of respiratory cell and molecular biology 20010401
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The allosteric interaction of otenzepad (AF-DX 116) at muscarinic M2 receptors in guinea pig atria.
European journal of pharmacology 20010330
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Gallamine triethiodide selectively blocks voltage-gated potassium channels in Ranvier nodes.
General physiology and biophysics 20010301
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Allosteric interactions of staurosporine and other indolocarbazoles with N-[methyl-(3)H]scopolamine and acetylcholine at muscarinic receptor subtypes: identification of a second allosteric site.
Molecular pharmacology 20000701
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Intubation conditions and postoperative myalgia in outpatient dental surgery: a comparison of succinylcholine with mivacurium.
Anaesthesia and intensive care 20000401
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The influence of peripheral site ligands on the reaction of symmetric and chiral organophosphates with wildtype and mutant acetylcholinesterases.
Chemico-biological interactions 19990514
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Myoclonic and tonic seizures elicited by microinjection of cholinergic drugs into the inferior colliculus.
Therapie 19990101
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Interaction of neuromuscular blocking drugs with recombinant human m1-m5 muscarinic receptors expressed in Chinese hamster ovary cells.
British journal of pharmacology 19981101
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Binding of the labelled muscarinic toxin 125I-MT1 to rat brain muscarinic M1 receptors.
European journal of pharmacology 19960603
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Assessment of the muscarinic receptor subtypes involved in pilocarpine-induced seizures in mice.
Neuroscience letters 19940227
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Adverse reaction to neuromuscular blockers: frequency, investigation, and epidemiology.
Acta anaesthesiologica Scandinavica. Supplementum 19940101
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The best prophylaxis for succinylcholine myalgias: extension of a previous meta-analysis.
Anesthesia and analgesia 19931101
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Ranitidine reverses gallamine paralysis in rats.
Anesthesia and analgesia 19930301
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Differential effects of neuromuscular blocking agents on suxamethonium-induced fasciculations and myalgia.
British journal of anaesthesia 19880301
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[Does diazepam prevent fasciculation and myalgias caused by suxamethonium? A double-blind study].
Ugeskrift for laeger 19870202
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Subclassification of muscarinic receptors in the heart, urinary bladder and sympathetic ganglia in the pithed rat. Selectivity of some classical agonists.
Naunyn-Schmiedeberg's archives of pharmacology 19851201
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Postoperative spasticity and shivering. A review with personal observations of 500 patients.
Anaesthesia 19840101
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Reduction of post-suxamethonium pain by pretreatment with four non-depolarizing agents.
British journal of anaesthesia 19810501
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Relation of precurarization to suxamethonium to provide ease of intubation and to prevent post-suxamethonium muscle pains.
Canadian Anaesthetists' Society journal 19790301
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Anesthesia related muscle paralysis in renal failure.
Clinical nephrology 19780701
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Comparative effects of nondepolarizing muscle relaxants on succinycholine-induced fasciculations and postoperative pain.
Southern medical journal 19770901
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The inhibitory effect of gallamine on muscarinic receptors.
British journal of pharmacology 19761101
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The effect of blood flow upon the activity of gallamine triethiodide.
British journal of anaesthesia 19760201
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Accidental subarachnoid injection of gallamine. A case report.
British journal of anaesthesia 19750801
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Comparison of gallamine with d-tubocurarine effects on fasciculations after succinylcholine.
Anesthesia and analgesia 19750101
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Accidental intrathecal injection of gallamine triethiodide.
Anaesthesia 19740501
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Cardiovascular collapse following succinylcholine in a paraplegic patient.
Paraplegia 19731101
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Quantitative aspects of the chronotropic and neuromuscular effects of gallamine in anesthetized man.
Anesthesiology 19711201
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Inhibition of succinylcholine-induced increased intragastric pressure by nondepolarizing muscle relaxants and lidocaine.
Anesthesiology 19710201
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Recurarization--fact or fiction.
Anesthesia and analgesia 19710101
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Analysis of anesthetic-related morbidity in human recipients of renal homografts.
Anesthesia and analgesia 19710101
