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Synthesis of some new benzisothiazolone and benzenesulfonamide derivatives of biological interest starting from saccharin sodium.
Archiv der Pharmazie 20131001
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Amide derivatives of benzene-sulfonanilide, pharmaceutical composition thereof and method for cancer treatment using the same (US20120095092).
Expert opinion on therapeutic patents 20121001
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Eight isostructural 4,4'-disubstituted N-phenylbenzenesulfonamides.
Acta crystallographica. Section C, Crystal structure communications 20121001
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Benzenesulfonamide attenuates monocrotaline-induced pulmonary arterial hypertension in a rat model.
European journal of pharmacology 20120905
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Virtual screening leads to the discovery of novel non-nucleotide P2Y₁ receptor antagonists.
Bioorganic & medicinal chemistry 20120901
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Placing supercritical fluid chromatography one step ahead of reversed-phase high performance liquid chromatography in the achiral purification arena: a hydrophilic interaction chromatography cross-linked diol chemistry as a new generic stationary phase.
Journal of chromatography. A 20120810
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Magnetic levitation as a platform for competitive protein-ligand binding assays.
Analytical chemistry 20120717
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FT-IR, FT-Raman and computational study of (E)-N-carbamimidoyl-4-((4-methoxybenzylidene)amino)benzenesulfonamide.
Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20120615
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Sulfonamide bearing oligonucleotides: simple synthesis and efficient RNA recognition.
Bioorganic & medicinal chemistry 20120615
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The novel endocrine disruptor tolylfluanid impairs insulin signaling in primary rodent and human adipocytes through a reduction in insulin receptor substrate-1 levels.
Biochimica et biophysica acta 20120601
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Research on the structure-surface adsorptive activity relationships of triazolyl glycolipid derivatives for mild steel in HCl.
Carbohydrate research 20120601
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Design of [(2-pyrimidinylthio)acetyl]benzenesulfonamides as inhibitors of human carbonic anhydrases.
European journal of medicinal chemistry 20120501
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N-(3-Methyl-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20120501
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N-(3-Nitro-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20120501
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Molecular cloning, characterization, and inhibition studies of a β-carbonic anhydrase from Malassezia globosa, a potential antidandruff target.
Journal of medicinal chemistry 20120412
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Discovery of novel 2-N-aryl-substituted benzenesulfonamidoacetamides: orally bioavailable tubulin polymerization inhibitors with marked antitumor activities.
ChemMedChem 20120401
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(3aR*,6S*,7aR*)-7a-Chloro-6-methyl-2-(4-methyl-phenyl-sulfon-yl)-2,3,3a,6,7,7a-hexa-hydro-3a,6-ep-oxy-1H-isoindole.
Acta crystallographica. Section E, Structure reports online 20120401
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Identification of novel kynurenine production-inhibiting benzenesulfonamide derivatives in cancer cells.
Biochemical and biophysical research communications 20120316
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Inhibitory effects of azole-type fungicides on interleukin-17 gene expression via retinoic acid receptor-related orphan receptors α and γ.
Toxicology and applied pharmacology 20120315
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Synthesis and evaluation of anticancer activity of some novel 6-aryl-2-(p-sulfamylphenyl)-pyridazin-3(2H)-ones.
European journal of medicinal chemistry 20120301
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4-{(4Z)-4-[(2Z)-3-(4-Fluoro-anilino)-1-hy-droxy-but-2-en-1-yl-idene]-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl}-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20120301
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Selective precipitation and purification of monovalent proteins using oligovalent ligands and ammonium sulfate.
Bioconjugate chemistry 20120215
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Synthesis and carbonic anhydrase inhibitory properties of novel cyclohexanonyl bromophenol derivatives.
Bioorganic & medicinal chemistry letters 20120201
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N-Ethyl-N-(4-methyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20120201
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2-(N-Cyclo-hexyl-carbamo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20120201
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Dependence of avidity on linker length for a bivalent ligand-bivalent receptor model system.
Journal of the American Chemical Society 20120111
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5-HT₂c receptor selectivity and structure-activity relationship of N-methyl-N-(1-methylpiperidin-4-yl)benzenesulfonamide analogs.
Bioorganic & medicinal chemistry letters 20120101
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Hydroxybenzothiazoles as new nonsteroidal inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1).
PloS one 20120101
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Novel 4-(4-substituted-thiazol-2-ylamino)-N-(pyridin-2-yl)-benzenesulfonamides as cytotoxic and radiosensitizing agents.
Archives of pharmacal research 20120101
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Synthesis, in-vitro anticancer screening and radiosensitizing evaluation of some new N-(quinoxalin-2-yl)benzenesulfonamide derivatives.
Arzneimittel-Forschung 20120101
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Regulation of expression of citrate synthase by the retinoic acid receptor-related orphan receptor α (RORα).
PloS one 20120101
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FH535 potentiation of cigarette smoke condensate cytotoxicity is associated with changes in β-catenin and EGR-1 signaling.
International journal of toxicology 20120101
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Label-free detection of protein binding with multisine SPR microchips.
Lab on a chip 20111221
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Estimation of analyte concentration by surface plasmon resonance-based biosensing using parameter identification techniques.
Analytical biochemistry 20111215
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FT-IR, FT-Raman and quantum chemical calculations of (E)-N-carbamimidoyl-4-((3,4-dimethoxybenzylidene) amino) benzenesulfonamide.
Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20111215
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Radiosynthesis of three [11C]ureido-substituted benzenesulfonamides as PET probes for carbonic anhydrase IX in tumors.
Bioorganic & medicinal chemistry letters 20111201
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Synthesis and biological evaluation of some new 2-pyrazolines bearing benzene sulfonamide moiety as potential anti-inflammatory and anti-cancer agents.
European journal of medicinal chemistry 20111201
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Synthesis, in vitro anticancer screening and radiosensitizing evaluation of some new 4-[3-(substituted)thioureido]-N-(quinoxalin-2-yl)-benzenesulfonamide derivatives.
Acta pharmaceutica (Zagreb, Croatia) 20111201
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Synthesis and acrosin inhibitory activity of substituted 4-amino-N-(diaminomethylene) benzenesulfonamide derivatives.
Bioorganic & medicinal chemistry letters 20111115
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A double prodrug system for colon targeting of benzenesulfonamide COX-2 inhibitors.
Bioorganic & medicinal chemistry letters 20111115
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Rhodium-catalyzed annulation of N-benzoylsulfonamide with isocyanide through C-H activation.
Chemistry (Weinheim an der Bergstrasse, Germany) 20111104
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Substituted phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonamides as antimitotics. Antiproliferative, antiangiogenic and antitumoral activity, and quantitative structure-activity relationships.
European journal of medicinal chemistry 20111101
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2,4-Dichloro-N-(3,5-dimethyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20111101
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4-Chloro-N-(3,4-dichloro-phen-yl)-2-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20111101
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Identification of novel small molecule inhibitors of 4-diphosphocytidyl-2-C-methyl-D-erythritol (CDP-ME) kinase of Gram-negative bacteria.
Bioorganic & medicinal chemistry 20111001
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Design and synthesis of new N-(5-trifluoromethyl)-1H-1,2,4-triazol-3-yl benzenesulfonamides as possible antimalarial prototypes.
Molecules (Basel, Switzerland) 20110920
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Synthesis of rhodamine B-benzenesulfonamide conjugates and their inhibitory activity against human α- and bacterial/fungal β-carbonic anhydrases.
Bioorganic & medicinal chemistry letters 20110915
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Fluoroalkyl and alkyl chains have similar hydrophobicities in binding to the 'hydrophobic wall' of carbonic anhydrase.
Journal of the American Chemical Society 20110907
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Synthesis and in vivo evaluation of [O-methyl-11C] N-[3,5-dichloro-2-(methoxy)phenyl]-4-(methoxy)-3-(1-piperazinyl)benzenesulfonamide as an imaging probe for 5-HT6 receptors.
Bioorganic & medicinal chemistry 20110901
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N-(2,6-Dimethyl-phen-yl)-2,4-dimethyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110901
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1-Benzyl-2,5-diphenyl-3-tosylimidazol-idin-4-one.
Acta crystallographica. Section E, Structure reports online 20110901
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4-(3-Methyl-5-phenyl-1H-pyrazol-1-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110901
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4-(3,7-Dimethyl-4-oxo-4,5-dihydro-isoxazolo[4,5-d]pyridazin-5-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110901
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4-(5-Oxo-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110901
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4-(3-Methyl-4,5-dihydro-1H-benzo[g]indazol-1-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110901
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Using covalent dimers of human carbonic anhydrase II to model bivalency in immunoglobulins.
Journal of the American Chemical Society 20110803
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Potassium N-bromo-2-methyl-benzene-sulfonamidate sesquihydrate.
Acta crystallographica. Section E, Structure reports online 20110801
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2-(4-Chloro-phen-yl)-5-(cyclo-hex-1-en-1-yl)-3-(4-methyl-phenyl-sulfon-yl)-1-phenyl-imidazolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20110801
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4-Chloro-N-(3,5-dimethyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110801
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Systematic errors in isothermal titration calorimetry: concentrations and baselines.
Analytical biochemistry 20110715
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Synthesis of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide as anticancer and anti-inflammatory agents.
Bioorganic & medicinal chemistry letters 20110715
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Potassium N,2-dichloro-benzene-sulfonamidate sesquihydrate.
Acta crystallographica. Section E, Structure reports online 20110701
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Potassium N,4-dichloro-benzene-sulfonamidate monohydrate.
Acta crystallographica. Section E, Structure reports online 20110701
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Potassium N-bromo-4-chloro-benzene-sulfonamidate monohydrate.
Acta crystallographica. Section E, Structure reports online 20110701
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Amino-caprolactam γ-secretase inhibitors showing potential for the treatment of Alzheimer's disease.
Bioorganic & medicinal chemistry letters 20110615
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Conformational variability of different sulfonamide inhibitors with thienyl-acetamido moieties attributes to differential binding in the active site of cytosolic human carbonic anhydrase isoforms.
Bioorganic & medicinal chemistry 20110615
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Crossing borders to bind proteins--a new concept in protein recognition based on the conjugation of small organic molecules or short peptides to polypeptides from a designed set.
Analytical and bioanalytical chemistry 20110601
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Ethyl 3-[2-(3,4-dimeth-oxy-benz-yl)-1-phenyl-sulfonyl-1H-indol-3-yl]acrylate chloro-form hemisolvate.
Acta crystallographica. Section E, Structure reports online 20110601
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A novel COX-2 inhibitor pyrazole derivative proven effective as an anti-inflammatory and analgesic drug.
Basic & clinical pharmacology & toxicology 20110401
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Synthesis and biological evaluation of some 4-functionalized-pyrazoles as antimicrobial agents.
European journal of medicinal chemistry 20110401
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2-(4-Chloro-phen-yl)-1,5-diphenyl-3-tosyl-imidazolidin-4-one.
Acta crystallographica. Section E, Structure reports online 20110401
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4-Chloro-N-(4-nitro-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110401
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2-Methyl-N-(4-nitro-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110401
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2-Chloro-N-(4-nitro-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110401
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Studies of tricyclic piperazine/piperidine furnished molecules as novel integrin αvβ3/αIIbβ3 dual antagonists using 3D-QSAR and molecular docking.
Journal of molecular graphics & modelling 20110201
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N-(4-Meth-oxy-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110201
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Molecular structure and vibrational investigation of benzenesulfonic acid methyl ester using DFT (LSDA, B3LYP, B3PW91 and MPW1PW91) theory calculations.
Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20110101
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Synthesis and in vitro anticancer evaluation of some novel hexahydroquinoline derivatives having a benzenesulfonamide moiety.
European journal of medicinal chemistry 20110101
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Correlation analyses on binding affinity of substituted benzenesulfonamides with carbonic anhydrase using ab initio MO calculations on their complex structures (II).
Bioorganic & medicinal chemistry letters 20110101
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Inhibition of β-carbonic anhydrases with ureido-substituted benzenesulfonamides.
Bioorganic & medicinal chemistry letters 20110101
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4-Chloro-N-(2,3-dichloro-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110101
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N-(2,5-Dichloro-phen-yl)-4-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110101
-
2,4-Dimethyl-N-(4-methyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20110101
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Induction of SCEs and DNA fragmentation in bovine peripheral lymphocytes by in vitro exposure to tolylfluanid-based fungicide.
Genetics and molecular biology 20110101
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Copper and its complexes in medicine: a biochemical approach.
Molecular biology international 20110101
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Virtual screening of 2,3-disubstituted-4(3H)-quinazolinones possessing benzenesulfonamide moiety for COX-2 inhibitor.
Bioinformation 20110101
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Inhibition of influenza A virus (H1N1) fusion by benzenesulfonamide derivatives targeting viral hemagglutinin.
PloS one 20110101
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Selective elution of target protein from affinity resins by a simple reductant with a thiol group.
Bioorganic & medicinal chemistry letters 20101215
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4- and 6-(p-Sulphamoylphenyl)androstenediones: Studies of aromatase inhibitor-based oestrone sulphatase inhibition.
Steroids 20101201
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Design and synthesis of an androgen receptor pure antagonist (CH5137291) for the treatment of castration-resistant prostate cancer.
Bioorganic & medicinal chemistry 20101201
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N-(2,3-Dichloro-phen-yl)-2,4-dimethyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20101201
-
N-(2,6-Dichloro-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20101201
-
N-(2,3-Dichloro-phen-yl)-4-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20101201
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N-(2,3-Dimethyl-phen-yl)-4-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20101201
-
5,6,7,8-Tetrahydropyrido[4,3-d]pyrimidines as novel class of potent and highly selective CaMKII inhibitors.
Bioorganic & medicinal chemistry letters 20101115
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A diverse series of substituted benzenesulfonamides as aldose reductase inhibitors with antioxidant activity: design, synthesis, and in vitro activity.
Journal of medicinal chemistry 20101111
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4-[N-(substituted 4-pyrimidinyl)amino]benzenesulfonamides as inhibitors of carbonic anhydrase isozymes I, II, VII, and XIII.
Bioorganic & medicinal chemistry 20101101
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Indapamide-like benzenesulfonamides as inhibitors of carbonic anhydrases I, II, VII, and XIII.
Bioorganic & medicinal chemistry 20101101
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Free-solution interaction assay of carbonic anhydrase to its inhibitors using back-scattering interferometry.
Electrophoresis 20101101
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N-(5-Chloro-2-meth-oxy-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20101101
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4-[(2-Hy-droxy-benzyl-idene)amino]-N-(5-methyl-isoxazol-3-yl)benzene-sulfonamide: a monoclinic polymorph.
Acta crystallographica. Section E, Structure reports online 20101001
-
Synthesis of anti-microtubule N-(2-Arylindol-7-yl)benzenesulfonamide derivatives and their antitumor mechanisms.
ChemMedChem 20100903
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Discovery of pyrrole-indoline-2-ones as Aurora kinase inhibitors with a different inhibition profile.
Journal of medicinal chemistry 20100826
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Identification of N-(2-(azepan-1-yl)-2-phenylethyl)-benzenesulfonamides as novel inhibitors of GlyT1.
Bioorganic & medicinal chemistry letters 20100815
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2-Methyl-N-(2-methyl-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100801
-
N-(4-Chloro-benzo-yl)-2-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100801
-
Cell adhesion to unnatural ligands mediated by a bifunctional protein.
Journal of the American Chemical Society 20100721
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Pteridine-sulfonamide conjugates as dual inhibitors of carbonic anhydrases and dihydrofolate reductase with potential antitumor activity.
Bioorganic & medicinal chemistry 20100715
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Coumarinyl-substituted sulfonamides strongly inhibit several human carbonic anhydrase isoforms: solution and crystallographic investigations.
Bioorganic & medicinal chemistry 20100715
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Synthesis of quinazolines from N-(2-nitrophenylsulfonyl)iminodiacetate and alpha-(2-nitrophenylsulfonyl)amino ketones via 2H-indazole 1-oxides.
The Journal of organic chemistry 20100702
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Synthesis and in vitro anticancer screening of some novel 4-[2-amino-3-cyano-4-substituted-5,6,7,8-tetrahydroquinolin-1-(4H)-yl]benzenesulfonamides.
European journal of medicinal chemistry 20100701
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2,4-Dichloro-N-(3-methyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100701
-
2,4-Dichloro-N-(3-chloro-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100701
-
N-(4-Methyl-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100701
-
New hydroxypyrimidinone-containing sulfonamides as carbonic anhydrase inhibitors also acting as MMP inhibitors.
Bioorganic & medicinal chemistry letters 20100615
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A rationale for the activity profile of benzenesulfonamide derivatives as cyclooxygenase (COX) inhibitors.
European journal of medicinal chemistry 20100601
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4-Chloro-N-(3,4-dimethyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100601
-
N-(Phenyl-sulfon-yl)acetamide.
Acta crystallographica. Section E, Structure reports online 20100601
-
2-Chloro-N-(3-chloro-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100601
-
2-Chloro-N-(4-methyl-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100601
-
Correlation analyses on binding affinity of substituted benzenesulfonamides with carbonic anhydrase using ab initio MO calculations on their complex structures.
Journal of chemical information and modeling 20100524
-
3D-QSAR study of benzene sulfonamide analogs as carbonic anhydrase II inhibitors.
Bioorganic & medicinal chemistry letters 20100515
-
Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: structure-based drug design, synthesis, and biological evaluation.
Bioorganic & medicinal chemistry 20100501
-
17,18-Dibromo-8-methyl-4,12-ditosyl-3,4,5,6,7,8,9,10,11,12,13,14-dodeca-hydro-2H-benzo[b][1,4,7,11,15]dioxatriaza-cyclo-hepta-decine.
Acta crystallographica. Section E, Structure reports online 20100501
-
N-Phenyl-N-(prop-2-en-1-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100501
-
N-(4-Hydroxy-phen-yl)benzene-sulfon-amide.
Acta crystallographica. Section E, Structure reports online 20100501
-
N-(3,5-Dichloro-phen-yl)-2,4-dimethyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100501
-
N-(2,6-Dimethyl-phen-yl)-4-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100501
-
catena-Poly[neodymium(III)-bis-[μ-N-(dimorpholinophosphor-yl)benzene-sulfonamidato]-sodium(I)-bis-[μ-N-(dimorpholinophosphor-yl)benzene-sulfonamidato]].
Acta crystallographica. Section E, Structure reports online 20100401
-
N-Cyclo-hexyl-4-meth-yl-N-propyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100401
-
2-Methyl-N-(4-methyl-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100401
-
2,4-Dimethyl-N-(3-methyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100401
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Recognition and binding of a helix-loop-helix peptide to carbonic anhydrase occurs via partly folded intermediate structures.
Biophysical journal 20100203
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N-(2-Chloro-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100201
-
N-(4-Chloro-benzo-yl)-4-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100201
-
2-Methyl-N-(3-methyl-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100201
-
cis-N-(2-Hydroxy-cyclo-hexyl)-p-toluene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100201
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Computational study of the interactions between guanine derivatives and cyclin-dependent kinase 2 (CDK2) by CoMFA and QM/MM.
Journal of chemical information and modeling 20100101
-
Synthesis and biological activities of some novel triazoloquinazolines and triazinoquinazolines containing benzenesulfonamide moieties.
Arzneimittel-Forschung 20100101
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Tamsulosin-induced severe hypotension during general anesthesia: a case report.
Journal of medical case reports 20100101
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Pharmacophore elucidation and molecular docking studies on 5-phenyl-1-(3-pyridyl)-1h-1,2,4-triazole-3-carboxylic acid derivatives as COX-2 inhibitors.
Scientia pharmaceutica 20100101
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[Synthesis and investigation on antidiabetic activity of 4-(1-aryl-3-oxo-5-phenylpentylamino) benzenesulfonamide].
Yao xue xue bao = Acta pharmaceutica Sinica 20100101
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N-Cyclo-hexyl-N-ethyl-4-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20100101
-
N,N'-Bis(phenyl-sulfon-yl)succinamide.
Acta crystallographica. Section E, Structure reports online 20100101
-
N,N'-Bis(phenyl-sulfon-yl)maleamide.
Acta crystallographica. Section E, Structure reports online 20100101
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Environmentally sensitive fluorescent sensors based on synthetic peptides.
Sensors (Basel, Switzerland) 20100101
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Radiolabelling of proteins with fluorine-18 via click chemistry.
Chemical communications (Cambridge, England) 20091228
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Thermodynamic optimisation in drug discovery: a case study using carbonic anhydrase inhibitors.
ChemMedChem 20091201
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N-Benzyl-N-cyclo-hexyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091201
-
4-Benzene-sulfonamido-benzoic acid.
Acta crystallographica. Section E, Structure reports online 20091201
-
N-Cyclo-hexyl-N-(prop-2-en-1-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091201
-
N-Benzyl-N-cyclo-hexyl-4-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091201
-
N-(4-Chloro-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091201
-
N-Cyclo-hexyl-N-propyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091201
-
4-Methyl-N-(2-methyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091201
-
Discovery and optimization of novel 4-[(aminocarbonyl)amino]-N-[4-(2-aminoethyl)phenyl]benzenesulfonamide ghrelin receptor antagonists.
Bioorganic & medicinal chemistry letters 20091101
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In vivo and in vitro anti-leishmanial activities of 4-nitro-N-pyrimidin- and N-pyrazin-2-ylbenzenesulfonamides, and N2-(4-nitrophenyl)-N1-propylglycinamide.
Bioorganic & medicinal chemistry 20091101
-
2,2-Dimethyl-N-(phenyl-sulfon-yl)acetamide.
Acta crystallographica. Section E, Structure reports online 20091101
-
N-(3-Chloro-benzo-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091101
-
N-(2,5-Dimethyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091101
-
N-Cyclohexyl-N-methylbenzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091101
-
Theoretical characterization of substrate access/exit channels in the human cytochrome P450 3A4 enzyme: involvement of phenylalanine residues in the gating mechanism.
The journal of physical chemistry. B 20091001
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N-Benzo-ylbenzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20091001
-
Carbonic anhydrase inhibitors. Inhibition of the Rv1284 and Rv3273 beta-carbonic anhydrases from Mycobacterium tuberculosis with diazenylbenzenesulfonamides.
Bioorganic & medicinal chemistry letters 20090901
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2-Chloro-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20090901
-
N-(2-Formyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20090901
-
N-(2-Acetyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20090901
-
o-Toluene-sulfonamide: a redetermination.
Acta crystallographica. Section E, Structure reports online 20090901
-
4-[(Z)-(2-Eth-oxy-4-oxochroman-3-yl-idene)methyl-amino]benzene-sulfonamide monohydrate.
Acta crystallographica. Section E, Structure reports online 20090801
-
2,4-Dichloro-N-(3,4-dichloro-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20090801
-
In vitro pharmacological characterization of a novel allosteric modulator of alpha 7 neuronal acetylcholine receptor, 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744), exhibiting unique pharmacological profile.
The Journal of pharmacology and experimental therapeutics 20090701
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Hybrid molecules between benzenesulfonamides and active antimicrobial benzo[d]isothiazol-3-ones.
European journal of medicinal chemistry 20090601
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Toward the development of metal-based synthetic nucleases: DNA binding and oxidative DNA cleavage of a mixed copper(II) complex with N-(9H-purin-6-yl)benzenesulfonamide and 1,10-phenantroline. Antitumor activity in human Caco-2 cells and Jurkat T lymphocytes. Evaluation of p53 and Bcl-2 proteins in the apoptotic mechanism.
Journal of inorganic biochemistry 20090601
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Sodium N-chloro-2-methyl-benzene-sulfonamidate sesquihydrate.
Acta crystallographica. Section E, Structure reports online 20090601
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4-Methyl-N-phenyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20090601
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Discovery of 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a novel positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor.
Journal of medicinal chemistry 20090528
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Investigation of the fate of sulfonamides downgradient of a decommissioned sewage farm near Berlin, Germany.
Journal of contaminant hydrology 20090512
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Ligand-directed tosyl chemistry for protein labeling in vivo.
Nature chemical biology 20090501
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Synthesis and biological evaluation of novel pyrazoles and pyrazolo[3,4-d]pyrimidines incorporating a benzenesulfonamide moiety.
Archiv der Pharmazie 20090401
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N-(3,4-Dimethyl-phen-yl)-4-methyl-benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20090401
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Addition reactions of chloro- or iodomethyllithium to imines. Synthesis of enantiopure aziridines and beta-chloroamines.
The Journal of organic chemistry 20090320
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Synthesis and biological evaluation of sulfonylurea and thiourea derivatives substituted with benzenesulfonamide groups as potential hypoglycemic agents.
Bioorganic & medicinal chemistry letters 20090315
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Improvement of monolithic solid material by utilization of spacer for identification of the target using affinity resins.
Bioorganic & medicinal chemistry letters 20090301
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Carbonic anhydrase inhibitors: two-prong versus mono-prong inhibitors of isoforms I, II, IX, and XII exemplified by photochromic cis-1,2-alpha-dithienylethene derivatives.
Bioorganic & medicinal chemistry letters 20090301
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Ethyl 2-[N-(2-Formyl-phen-yl)benzene-sulfonamido]acetate.
Acta crystallographica. Section E, Structure reports online 20090301
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A novel class of allosteric modulators of AMPA/Kainate receptors.
Bioorganic & medicinal chemistry letters 20090215
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Synthesis and biological evaluation of benzenesulfonamide-substituted 4-(6-alkylpyridin-2-yl)-5-(quinoxalin-6-yl)imidazoles as transforming growth factor-beta type 1 receptor kinase inhibitors.
European journal of medicinal chemistry 20090201
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Synthesis of some pyrazolyl benzenesulfonamide derivatives as dual anti-inflammatory antimicrobial agents.
Journal of enzyme inhibition and medicinal chemistry 20090201
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N-(2,3-Dimethyl-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20090201
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Cryptophane xenon-129 nuclear magnetic resonance biosensors targeting human carbonic anhydrase.
Journal of the American Chemical Society 20090121
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Synthesis and antiinflammatory activity of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide.
Bioorganic & medicinal chemistry letters 20090101
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Label-free determination of protein-ligand binding constants using mass spectrometry and validation using surface plasmon resonance and isothermal titration calorimetry.
Journal of molecular recognition : JMR 20090101
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Synthesis and Antiviral Studies of Novel N-Sulphonamidomethyl piperazinyl Fluoroquinolones.
Indian journal of pharmaceutical sciences 20090101
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Dual inhibitors of matrix metalloproteinases and carbonic anhydrases: iminodiacetyl-based hydroxamate-benzenesulfonamide conjugates.
Journal of medicinal chemistry 20081225
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Synthesis of biologically active N-methyl derivatives of amidines and cyclized five-membered products of amidines with oxalyl chloride.
European journal of medicinal chemistry 20081201
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Recent improvements in the development of A(2B) adenosine receptor agonists.
Purinergic signalling 20081201
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Effect of the oral absorption of benzenesulfonanilide-type cyclooxygenase-1 inhibitors on analgesic action and gastric ulcer formation.
Journal of pharmaceutical sciences 20081201
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N-(3,5-Dichloro-phen-yl)benzene-sulfonamide.
Acta crystallographica. Section E, Structure reports online 20081101
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External pH influences the transcriptional profile of the carbonic anhydrase, CAH-4b in Caenorhabditis elegans.
Molecular and biochemical parasitology 20081001
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Tetra-aquabis-(2-sulfamoylbenzoato)manganese(II).
Acta crystallographica. Section E, Structure reports online 20081001
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Residual ligand entropy in the binding of p-substituted benzenesulfonamide ligands to bovine carbonic anhydrase II.
Journal of the American Chemical Society 20080917
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Chromofluorescent indicator for intracellular Zn2+/Hg2+ dynamic exchange.
Organic letters 20080904
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Photophysical and complexation properties of benzenesulfonamide derivatives with different donor and acceptor moieties.
Journal of fluorescence 20080901
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Tetramethylcyclopropyl analogue of the leading antiepileptic drug, valproic acid: evaluation of the teratogenic effects of its amide derivatives in NMRI mice.
Birth defects research. Part A, Clinical and molecular teratology 20080901
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Chemometrical examination of active parameters and interactions in flow injection-capillary electrophoresis.
Electrophoresis 20080901
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Inhibition of human mitochondrial carbonic anhydrases VA and VB with para-(4-phenyltriazole-1-yl)-benzenesulfonamide derivatives.
Bioorganic & medicinal chemistry letters 20080815
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2,2,2-Trimethyl-N-(phenyl-sulfon-yl)-acetamide.
Acta crystallographica. Section E, Structure reports online 20080801
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2,2-Dichloro-N-(phenyl-sulfon-yl)-acetamide.
Acta crystallographica. Section E, Structure reports online 20080801
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Affinity-labeling-based introduction of a reactive handle for natural protein modification.
Chemistry, an Asian journal 20080707
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Carbonic anhydrase inhibitors: design of spin-labeled sulfonamides incorporating TEMPO moieties as probes for cytosolic or transmembrane isozymes.
Bioorganic & medicinal chemistry letters 20080615
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Exploration of physicochemical properties and molecular modelling studies of 2-sulfonyl-phenyl-3-phenyl-indole analogs as cyclooxygenase-2 inhibitors.
European journal of medicinal chemistry 20080601
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Similar sulfonamides with different crystal structures: sulfasymazine and sulfatriazine.
Acta crystallographica. Section C, Crystal structure communications 20080601
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Antidiabetic activity of N-(6-substituted-1,3-benzothiazol-2-yl)benzenesulfonamides.
Bioorganic & medicinal chemistry letters 20080501
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2-[N-(X-chlorophenyl)carbamoyl]benzenesulfonamide (with X = 2 and 4).
Acta crystallographica. Section C, Crystal structure communications 20080501
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Functional human 5-HT6 receptor assay for high throughput screening of chemical ligands and binding proteins.
Combinatorial chemistry & high throughput screening 20080501
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Behaviour and biodegradation of sulfonamides (p-TSA, o-TSA, BSA) during drinking water treatment.
Chemosphere 20080401
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Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides.
Bioorganic & medicinal chemistry 20080401
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Design and synthesis of N-(3,5-difluoro-4-hydroxyphenyl)benzenesulfonamides as aldose reductase inhibitors.
Bioorganic & medicinal chemistry 20080401
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Electrophysiological characterization of a novel Kv channel blocker N,N'-[oxybis(2,1-ethanediyloxy-2,1-ethanediyl) ]bis(4-methyl)-benzenesulfonamide found in virtual screening.
Acta pharmacologica Sinica 20080401
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Ethyl 2-(bromo-meth-yl)-5-meth-oxy-1-phenyl-sulfonyl-1H-indole-3-carboxyl-ate.
Acta crystallographica. Section E, Structure reports online 20080401
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Identification and significance of sulphonamides (p-TSA, o-TSA, BSA) in an urban water cycle (Berlin, Germany).
Water research 20080301
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Selective COX-2 inhibitors. Part 2: synthesis and biological evaluation of 4-benzylideneamino- and 4-phenyliminomethyl-benzenesulfonamides.
Bioorganic & medicinal chemistry 20080301
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Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: Effect of the N-5 bond type on the affinity and selectivity at the four adenosine receptor subtypes.
Purinergic signalling 20080301
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Synthesis and cyclooxygenase inhibitory activities of linear 1-(methanesulfonylphenyl or benzenesulfonamido)-2-(pyridyl)acetylene regioisomers.
Bioorganic & medicinal chemistry 20080215
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Benzenesulfonamide indole inhibitors of cytosolic phospholipase A2alpha: optimization of in vitro potency and rat pharmacokinetics for oral efficacy.
Bioorganic & medicinal chemistry 20080201
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Metal-based sulfonamides: their preparation, characterization and in-vitro antibacterial, antifungal & cytotoxic properties. X-ray structure of 4-[(2-hydroxybenzylidene) amino] benzenesulfonamide.
Journal of enzyme inhibition and medicinal chemistry 20080201
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Ethyl 2-[(phenyl-sulfan-yl)meth-yl]-1-(phenyl-sulfon-yl)-1H-indole-3-carboxyl-ate.
Acta crystallographica. Section E, Structure reports online 20080201
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(2-Methyl-1-phenyl-sulfonyl-1H-indol-3-yl)methanol.
Acta crystallographica. Section E, Structure reports online 20080201
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Carbonic anhydrase inhibitors: copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII.
Bioorganic & medicinal chemistry letters 20080115
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New celecoxib derivatives as anti-inflammatory agents.
Journal of medicinal chemistry 20080110
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Identification of N-(quinolin-8-yl)benzenesulfonamides as agents capable of down-regulating NFkappaB activity within two separate high-throughput screens of NFkappaB activation.
Bioorganic & medicinal chemistry letters 20080101
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An efficient solvent-free synthesis of benzoxanthenes catalyzed by BSA or O-TSA.
Preparative biochemistry & biotechnology 20080101
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Antimicrobial activity of some sulfonamide derivatives on clinical isolates of Staphylococus aureus.
Annals of clinical microbiology and antimicrobials 20080101
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Binding modes of two novel non-nucleoside reverse transcriptase inhibitors, YM-215389 and YM-228855, to HIV type-1 reverse transcriptase.
Antiviral chemistry & chemotherapy 20080101
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Small molecule inhibitors of integrin alpha2beta1.
Journal of medicinal chemistry 20071101
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A remarkable accelerating effect of Ag-salt on intramolecular cyclization of o-(1-alkynyl)benzenesulfonamides.
The Journal of organic chemistry 20071026
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A strategy for designing 'multi-prong' enzyme inhibitors by incorporating selective ligands to the liposomal surface.
Chemical communications (Cambridge, England) 20070828
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Design, synthesis and pharmacological evaluation of 4-[2-alkylthio-5(4)-(4-substitutedphenyl)imidazole-4(5)yl]benzenesulfonamides as selective COX-2 inhibitors.
Acta pharmacologica Sinica 20070801
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Quantitative determination of three sulfonamides in environmental water samples using liquid chromatography coupled to electrospray tandem mass spectrometry.
Journal of chromatography. A 20070720
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Structure-based design of 2-arylamino-4-cyclohexylmethoxy-5-nitroso-6-aminopyrimidine inhibitors of cyclin-dependent kinase 2.
Organic & biomolecular chemistry 20070521
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Structural analysis of charge discrimination in the binding of inhibitors to human carbonic anhydrases I and II.
Journal of the American Chemical Society 20070502
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Pharmacophoric 2-hydroxyalkyl benzenesulfonamide: a single-step synthesis from benzenesulfonamide via hemiaminal.
European journal of medicinal chemistry 20070401
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Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated isoforms I, II, and IX with iminodiacetic carboxylates/hydroxamates also incorporating benzenesulfonamide moieties.
Bioorganic & medicinal chemistry letters 20070315
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Synthesis and in vivo evaluation of [18F]-4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide as a PET imaging probe for COX-2 expression.
Bioorganic & medicinal chemistry 20070215
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Dependence of effective molarity on linker length for an intramolecular protein-ligand system.
Journal of the American Chemical Society 20070207
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Thermodynamic parameters for the association of fluorinated benzenesulfonamides with bovine carbonic anhydrase II.
Chemistry, an Asian journal 20070108
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Strategies for controlled placement of nanoscale building blocks.
Nanoscale research letters 20070101
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Discovery of HIV-1 protease inhibitors with picomolar affinities incorporating N-aryl-oxazolidinone-5-carboxamides as novel P2 ligands.
Journal of medicinal chemistry 20061214
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Thiol-mediated anchoring of ligands to self-assembled monolayers for studies of biospecific interactions.
Langmuir : the ACS journal of surfaces and colloids 20061121
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Synthesis and in vitro antitumor evaluation of some indeno[1,2-c]pyrazol(in)es substituted with sulfonamide, sulfonylurea(-thiourea) pharmacophores, and some derived thiazole ring systems.
Bioorganic & medicinal chemistry 20061001
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Intracellular inhibition of carboxylesterases by benzil: modulation of CPT-11 cytotoxicity.
Molecular cancer therapeutics 20060901
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Binding of sulfonyl-containing arylalkylamines at human 5-HT6 serotonin receptors.
Journal of medicinal chemistry 20060824
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Urotensin-II blockade with SB-611812 attenuates cardiac dysfunction in a rat model of coronary artery ligation.
Journal of molecular and cellular cardiology 20060801
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Sorption-desorption of flucarbazone and propoxycarbazone and their benzenesulfonamide and triazolinone metabolites in two soils.
Pest management science 20060701
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Carbonic anhydrase inhibitors: cloning and sulfonamide inhibition studies of a carboxyterminal truncated alpha-carbonic anhydrase from Helicobacter pylori.
Bioorganic & medicinal chemistry letters 20060415
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Molecular structure and conformations of benzenesulfonamide: gas electron diffraction and quantum chemical calculations.
The Journal of organic chemistry 20060414
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Benzoxazole benzenesulfonamides are novel allosteric inhibitors of fructose-1,6-bisphosphatase with a distinct binding mode.
Bioorganic & medicinal chemistry letters 20060401
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Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs.
Journal of medicinal chemistry 20060323
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Ultrahigh resolution crystal structures of human carbonic anhydrases I and II complexed with 'two-prong' inhibitors reveal the molecular basis of high affinity.
Journal of the American Chemical Society 20060308
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Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II 'selective' inhibitor celecoxib.
Bioorganic & medicinal chemistry letters 20060115
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Downregulation of survivin expression and concomitant induction of apoptosis by celecoxib and its non-cyclooxygenase-2-inhibitory analog, dimethyl-celecoxib (DMC), in tumor cells in vitro and in vivo.
Molecular cancer 20060101
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Short communication inhibitory activity of 4-[(1,2-dihydro-2-oxo-3H-indol-3-ylidene)amino]-N-(4,6-dimethylpyrimidin-2-yl) benzenesulphonamide and its derivatives against orthopoxvirus replication in vitro.
Antiviral chemistry & chemotherapy 20060101
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CC 05, a novel anti-inflammatory compound, exerts its effect by inhibition of cyclooxygenase-2 activity.
European journal of pharmacology 20050927
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QSAR analysis of thiazole benzenesulfonamide substituted 3-pyridylethanolamines as beta3-adrenergic receptor agonist.
Bioorganic & medicinal chemistry letters 20050615
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Carbonic anhydrase inhibitors. Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with Schiff's bases incorporating chromone and aromatic sulfonamide moieties, and their zinc complexes.
Bioorganic & medicinal chemistry letters 20050615
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Synthesis and biological evaluation of 3,4-diphenyl-1,2,5-oxadiazole-2-oxides and 3,4-diphenyl-1,2,5-oxadiazoles as potential hybrid COX-2 inhibitor/nitric oxide donor agents.
Bioorganic & medicinal chemistry 20050415
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Design, synthesis, and biological evaluation of N-acetyl-2-carboxybenzenesulfonamides: a novel class of cyclooxygenase-2 (COX-2) inhibitors.
Bioorganic & medicinal chemistry 20050401
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Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II.
Bioorganic & medicinal chemistry letters 20050401
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Benzenesulfonamide analogs of fluoroquinolones. Antibacterial activity and QSAR studies.
European journal of medicinal chemistry 20050401
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Discovery and selection of TMC114, a next generation HIV-1 protease inhibitor.
Journal of medicinal chemistry 20050324
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Spacer-based selectivity in the binding of 'two-prong' ligands to recombinant human carbonic anhydrase I.
Biochemistry 20050308
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Studies of non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: synthesis and structure-activity relationships of 2-cyano and 2-hydroxy thiazolidenebenzenesulfonamide derivatives.
Bioorganic & medicinal chemistry 20050215
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QSAR studies on benzene sulfonamide carbonic anhydrase inhibitors: need of hydrophobic parameter for topological modeling of binding constants of sulfonamides to human CA-II.
Bioorganic & medicinal chemistry letters 20050215
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Novel use of chemical shift in NMR as molecular descriptor: a first report on modeling carbonic anhydrase inhibitory activity and related parameters.
Bioorganic & medicinal chemistry letters 20050215
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Characterization of beta3-adrenergic receptor: determination of pharmacophore and 3D QSAR model for beta3 adrenergic receptor agonism.
Journal of computer-aided molecular design 20050201
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Predictive flip regression: a technique for QSAR of derivatives of symmetric molecules.
Journal of chemical information and modeling 20050101
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In situ click chemistry: enzyme-generated inhibitors of carbonic anhydrase II.
Angewandte Chemie (International ed. in English) 20041217
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Studies of nonnucleoside HIV-1 reverse transcriptase inhibitors. Part 1: Design and synthesis of thiazolidenebenzenesulfonamides.
Bioorganic & medicinal chemistry 20041201
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Pharmacomodulation of a sulfamide 5-HT6 receptor ligand.
Journal of enzyme inhibition and medicinal chemistry 20041201
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Topological modeling of lipophilicity, diuretic activity, and carbonic inhibition activity of benzene sulfonamides: a molecular connectivity approach.
Bioorganic & medicinal chemistry letters 20041115
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Carbonic anhydrase inhibitors: inhibition of human cytosolic isozyme II and mitochondrial isozyme V with a series of benzene sulfonamide derivatives.
Bioorganic & medicinal chemistry letters 20041115
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Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties.
Bioorganic & medicinal chemistry letters 20041101
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Two-prong inhibitors for human carbonic anhydrase II.
Journal of the American Chemical Society 20041020
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Novel synthesis of 3,4-diarylisoxazole analogues of valdecoxib: reversal cyclooxygenase-2 selectivity by sulfonamide group removal.
Journal of medicinal chemistry 20040923
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Protein surface-assisted enhancement in the binding affinity of an inhibitor for recombinant human carbonic anhydrase-II.
Journal of the American Chemical Society 20040908
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Synthesis and antiviral activity of P1' arylsulfonamide azacyclic urea HIV protease inhibitors.
Bioorganic & medicinal chemistry letters 20040802
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Synthesis, antiviral, and anti-HIV-1 integrase activities of 3-aroyl-1,1-dioxo-1,4,2-benzodithiazines.
Bioorganic & medicinal chemistry 20040701
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Rewiring cell adhesion.
Journal of the American Chemical Society 20040602
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A versatile polypeptide platform for integrated recognition and reporting: affinity arrays for protein-ligand interaction analysis.
Chemistry (Weinheim an der Bergstrasse, Germany) 20040517
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New heteroarylbenzenesulphonamides as matrix metalloproteinase inhibitors.
Bioorganic & medicinal chemistry letters 20040308
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Abeta aggregation inhibitors. Part 1: Synthesis and biological activity of phenylazo benzenesulfonamides.
Bioorganic & medicinal chemistry letters 20040308
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QSAR study on benzenesulphonamide carbonic anhydrase inhibitors: topological approach using Balaban index.
Bioorganic & medicinal chemistry 20040215
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Polar substitutions in the benzenesulfonamide ring of celecoxib afford a potent 1,5-diarylpyrazole class of COX-2 inhibitors.
Bioorganic & medicinal chemistry letters 20040119
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Application of CoMFA and CoMSIA 3D-QSAR and docking studies in optimization of mercaptobenzenesulfonamides as HIV-1 integrase inhibitors.
Journal of medicinal chemistry 20040115
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QSAR study using topological indices for inhibition of carbonic anhydrase II by sulfanilamides and Schiff bases.
Molecular diversity 20040101
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Synthesis and cyclooxygenase-2 inhibiting property of 1,5-diarylpyrazoles with substituted benzenesulfonamide moiety as pharmacophore: Preparation of sodium salt for injectable formulation.
Journal of medicinal chemistry 20030911
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Sorption-desorption of two 'aged' sulfonylaminocarbonyltriazolinone herbicide metabolites in soil.
Journal of agricultural and food chemistry 20030604
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Synthesis of 1-(6-chloro-1,1-dioxo-1,4,2-benzodithiazin-3-yl)semi-carbazides and their transformation into 4-chloro-2-mercapto-N-(4,5-dihydro-5-oxo-4-phenyl-1H-1,2,4-triazol-3-yl)benzenesulfonamides as potential anticancer and anti-HIV agents.
Farmaco (Societa chimica italiana : 1989) 20030601
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Valdecoxib-induced toxic epidermal necrolysis in a patient allergic to sulfa drugs.
Pharmacotherapy 20030401
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Tripodal ligand incorporating dual fluorescent ionophore: a coordinative control of photoinduced electron transfer.
Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology 20030301
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Synthesis of heteroaromatic analogues of (2-aryl-1-cyclopentenyl-1-alkylidene)-(arylmethyloxy)amine COX-2 inhibitors: effects on the inhibitory activity of the replacement of the cyclopentene central core with pyrazole, thiophene or isoxazole ring.
European journal of medicinal chemistry 20030201
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Using cyclooxygenase-2 inhibitors as molecular platforms to develop a new class of apoptosis-inducing agents.
Journal of the National Cancer Institute 20021204
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Diversity in the oxidation of substrates by cytochrome P450 2D6: lack of an obligatory role of aspartate 301-substrate electrostatic bonding.
Biochemistry 20020910
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An excretion balance and pharmacokinetic study of the novel anticancer agent E7070 in cancer patients.
Anti-cancer drugs 20020901
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The pharmacokinetics of a thiazole benzenesulfonamide beta 3-adrenergic receptor agonist and its analogs in rats, dogs, and monkeys: improving oral bioavailability.
Drug metabolism and disposition: the biological fate of chemicals 20020701
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Metabolism of a thiazole benzenesulfonamide derivative, a potent and elective agonist of the human beta3-adrenergic receptor, in rats: identification of a novel isethionic acid conjugate.
Drug metabolism and disposition: the biological fate of chemicals 20020701
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Effects of soil pH and soil water content on prosulfuron dissipation.
Journal of agricultural and food chemistry 20020522
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Enantiomeric separation of a thiazolbenzenesulfonamide compound using packed-column subcritical fluid chromatography.
Chirality 20020515
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Synthesis of unsymmetrical aroyl acyl imides by aminocarbonylation of aryl bromides.
The Journal of organic chemistry 20020125
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Rational determination of transfer free energies of small drugs across the water-oil interface.
Journal of medicinal chemistry 20020103
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Synthesis, characterization and antifungal activities of some benzenesulphonylamino acid derivatives.
Bollettino chimico farmaceutico 20020101
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Synthesis and anti-HIV activity of 4-[(1,2-dihydro-2-oxo-3H-indol-3-ylidene) amino]-N(4,6-dimethyl-2-pyrimidinyl)-benzene sulfonamide and its derivatives.
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20011201
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Comparative study of new benzenesulphonamide fluoroquinolones structurally related to ciprofloxacin against selected ciprofloxacin-susceptible and -resistant Gram-positive cocci.
The Journal of antimicrobial chemotherapy 20011101
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Subtle differences in dissociation rates of interactions between destabilized human carbonic anhydrase II mutants and immobilized benzenesulfonamide inhibitors probed by a surface plasmon resonance biosensor.
Analytical biochemistry 20010915
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Two isomorphous benzenesulfonamide crystal structures determined by intermolecular C-H...O, C-H...pi and C-H...Cl interactions.
Acta crystallographica. Section C, Crystal structure communications 20010901
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Synthesis of optically active N-(2-pyridyloxiran-2-ylmethyl) benzenesulfonamide derivatives and their herbicidal activity.
Bioscience, biotechnology, and biochemistry 20010701
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Ethenesulfonamide derivatives, a novel class of orally active endothelin-A receptor antagonists.
Chemical & pharmaceutical bulletin 20010501
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QSAR of antineoplastics IV: Hansch analysis of N-(7-indolyl)benzenesulfonamides against KB human nasopharynx carcinoma, colon 38 murine adenocarcinoma and P388 murine leukemia cell lines.
Drug design and discovery 20010101
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QSAR of antineoplastics V: Exploration of receptor interaction sites of antitumor N-(7-indolyl)benzenesulfonamides targeting GI phase using electrotopological state atom index.
Drug design and discovery 20010101
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Design and synthesis of benzoic acid derivatives as influenza neuraminidase inhibitors using structure-based drug design.
Journal of medicinal chemistry 19971205